SCHEMBL2917896

SCHEMBL2917896

C#CCNC(=O)c1cccc(F)c1Nc1nc(Nc2ccc3c(c2)OCCCN3CC)ncc1Cl.C#CCNC(=O)c1cccc(F)c1Nc1nc(Nc2ccc3c(c2)OCCCN3CC)ncc1Cl

nearest known ligand 0.83

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
MET P08581 20/20 0.83
INSR P06213 19/20 0.83

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL884909 1.00 MET (0.83) METINSR
SCHEMBL886723 0.92 MET (0.84) METINSR
SCHEMBL885070 0.91 MET (1.00) METINSR
SCHEMBL885323 0.91 MET (0.82) METINSR
SCHEMBL884973 0.90 MET (0.83) METINSR
SCHEMBL886223 0.88 MET (0.84) METINSR
SCHEMBL2063218 0.87 MET (0.83) METINSR
SCHEMBL2914471 0.87 MET (0.77) METINSR
SCHEMBL885077 0.87 MET (0.85) METINSR
SCHEMBL885309 0.87 MET (0.82) METINSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2222647-A1 FUSED BICYCLIC DERIVATIVES OF 2,4-DIAMINOPYRIMIDINE AS ALK AND C-MET INHIBITORS Cephalon, Inc. (US) 2010-09-01 EP disclosed
WO-2008051547-A1 FUSED BICYCLIC DERIVATIVES OF 2,4-DIAMINOPYRIMIDINE AS ALK AND C-MET INHIBITORS CEPHALON, INC. (US) 2008-05-02 WO disclosed