SCHEMBL2918059

SCHEMBL2918059

CSc1cccc2c1C(=O)N(c1ccc(C(F)(C(F)(F)F)C(F)(F)F)cc1C)C2=O

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
GRM1 Q13255 8/20 0.38
GRM4 Q14833 8/20 0.38
TYMS P04818 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
DPP4 P27487 1/20 0.36
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2916208 0.84 GRM1 (0.52) LMNASMN1; SMN2GRM1GRM4
SCHEMBL5418153 0.83 LMNA (0.42) LMNASMN1; SMN2GRM1GRM4TYMS
SCHEMBL3374587 0.83 ANPEP (0.46) LMNASMN1; SMN2GRM1GRM4TYMS
SCHEMBL5429466 0.83 GRM1 (0.51) LMNASMN1; SMN2GRM1GRM4
SCHEMBL2916938 0.81 LMNA (0.40) LMNASMN1; SMN2GRM1GRM4TYMS
SCHEMBL3376357 0.78 LMNA (0.47) LMNASMN1; SMN2GRM1GRM4TYMS
SCHEMBL3376337 0.77 LMNA (0.46) LMNASMN1; SMN2GRM1GRM4TYMS
SCHEMBL3376240 0.76 LMNA (0.45) LMNASMN1; SMN2GRM1GRM4TYMS
SCHEMBL14579468 0.74 GRM1 (0.41) LMNASMN1; SMN2GRM1GRM4MEN1
SCHEMBL12402290 0.74 HPGD (0.35) LMNASMN1; SMN2GRM1GRM4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1006107-B1 Phthalamide derivatives, or salt thereof agrohorticultural insecticide, and method for using the same NIHON NOHYAKU CO LTD (JP) 2010-09-01 EP disclosed
US-6603044-B1 The present invention provides a phthalamide derivative of the formula (I): agrohorticultural insecticide containing said compound as active ingredient and exhibiting an excellent insecticidal effect. NIHON NOHYAKU CO., LTD. (JP) 2003-08-05 US disclosed
EP-1006107-A2 Phthalamide derivatives, or salt thereof agrohorticultural insecticide, and method for using the same NIHON NOHYAKU CO., LTD. (JP) 2000-06-07 EP disclosed