SCHEMBL29189474

SCHEMBL29189474

COC(=O)c1ccc(NC(=O)O)c(OC2CC2)c1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 3/20 0.46
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
PDE4D Q08499 5/20 0.45
PDE4A P27815 4/20 0.45
PDE4B Q07343 4/20 0.45
PDE4C Q08493 4/20 0.45
EPHX2 P34913 1/20 0.44
HSP90AB1 P08238 2/20 0.44
TOP2A P11388 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
PYGL P06737 1/20 0.44
ALOX15 P16050 1/20 0.43
NOTUM Q6P988 1/20 0.43
MAPT P10636 1/20 0.42
PDE1A P54750 1/20 0.42
PDE1B Q01064 1/20 0.42
PDE1C Q14123 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29189691 0.88 PDE4B (0.44) PDE5AKDM4EALDH1A1PDE4DPDE4A
SCHEMBL23958622 0.83 PDE5A (0.43) PDE5AKDM4EALDH1A1PDE4DPDE4A
SCHEMBL30117191 0.82 NOTUM (0.54) PDE5AKDM4EALDH1A1PDE4DPDE4A
SCHEMBL23704079 0.82 NOTUM (0.54) PDE5AKDM4EALDH1A1PDE4DPDE4A
SCHEMBL24751982 0.82 EPHX2 (0.44) PDE5AKDM4EALDH1A1PDE4DPDE4A
SCHEMBL30138077 0.82 EPHX2 (0.44) PDE5AKDM4EALDH1A1PDE4DPDE4A
SCHEMBL18031253 0.82 MAPT (0.53) PDE5APDE4DPDE4APDE4BPDE4C
SCHEMBL16544967 0.80 MAPT (0.62) PDE5APDE4DPDE4APDE4BPDE4C
SCHEMBL18031244 0.80 CA12 (0.57) PDE5AKDM4EALDH1A1PDE4DPDE4A
SCHEMBL29208134 0.79 ALDH1A1 (0.42) PDE5AKDM4EALDH1A1PDE4DPDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117881681-A Substituted pyrrolo [2,3-d ] pyrimidines, their preparation and their therapeutic use 赛诺菲 2024-04-12 CN disclosed