SCHEMBL29196400

SCHEMBL29196400

ON1CC[CH]C1CCc1ccc2ccccc2c1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 4/20 0.47
SLC6A4 P31645 1/20 0.43
CYP1A2 P05177 1/20 0.43
KMT2A Q03164 1/20 0.41
SIGMAR1 Q99720 3/20 0.41
ACHE P22303 1/20 0.40
PKM P14618 1/20 0.40
HDAC3 O15379 2/20 0.40
HDAC4 P56524 2/20 0.40
HDAC1 Q13547 2/20 0.40
HDAC7 Q8WUI4 2/20 0.40
HDAC2 Q92769 2/20 0.40
HDAC10 Q969S8 2/20 0.40
HDAC11 Q96DB2 2/20 0.40
HDAC8 Q9BY41 2/20 0.40
HDAC6 Q9UBN7 2/20 0.40
HDAC9 Q9UKV0 2/20 0.40
HDAC5 Q9UQL6 2/20 0.40
NAAA Q02083 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29196396 0.74 SLC18A2 (0.48) HRH3SLC6A4SIGMAR1ACHEHDAC3
SCHEMBL29196393 0.72 HRH3 (0.44) HRH3SLC6A4CYP1A2KMT2ASIGMAR1
SCHEMBL8669331 0.70 BCHE (0.51) HRH3SLC6A4CYP1A2KMT2ASIGMAR1
SCHEMBL29560700 0.68 CYP1A2 (0.65) HRH3SLC6A4CYP1A2KMT2ASIGMAR1
SCHEMBL6240981 0.68 CYP1A2 (0.65) HRH3SLC6A4CYP1A2KMT2ASIGMAR1
SCHEMBL8669223 0.67 BCHE (0.59) HRH3SLC6A4CYP1A2SIGMAR1ACHE
SCHEMBL6942749 0.67 HRH3 (0.47) HRH3SLC6A4CYP1A2KMT2ASIGMAR1
SCHEMBL9877336 0.67 HCRTR1 (0.45) HRH3SLC6A4CYP1A2ACHENAAA
SCHEMBL1581891 0.67 GRIN2D (0.50) HRH3CYP1A2SIGMAR1ACHE
SCHEMBL79723 0.65 CYP1A2 (0.56) HRH3SLC6A4CYP1A2SIGMAR1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117924217-A 5-HTT/HDAC dual inhibitor and preparation method and application thereof 杭州师范大学 2024-04-26 CN disclosed