SCHEMBL29196807

SCHEMBL29196807

CC(C)(C)P(Pc1ccnn1-c1c(-c2ccccc2)nn(-c2ccccc2)c1-c1ccccc1)C(C)(C)C

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.35
CA2 P00918 4/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
CCNA2 P20248 2/20 0.33
CDK2 P24941 2/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33
PTGS2 P35354 3/20 0.32
PTGS1 P23219 2/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
POLB P06746 1/20 0.32
MDM2 Q00987 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL140011 0.80 CA1 (0.37) CA1CA2MEN1KMT2ACYP1A2
SCHEMBL12930022 0.76 CYP2C9 (0.43) CA1CA2MEN1KMT2ACYP1A2
SCHEMBL11998814 0.76 CA1 (0.34) CA1CA2MEN1KMT2ACYP1A2
SCHEMBL28924190 0.76 MEN1 (0.36) CA1CA2MEN1KMT2ACYP1A2
SCHEMBL18806835 0.75 CA1 (0.37) CA1CA2MEN1KMT2ACYP1A2
SCHEMBL18802300 0.75 CA1 (0.37) CA1CA2MEN1KMT2ACYP1A2
SCHEMBL409808 0.74 CA1 (0.41) CA1CA2MEN1KMT2ACYP1A2
SCHEMBL28599216 0.74 MEN1 (0.37) CA1CA2MEN1KMT2ACYP1A2
SCHEMBL1332907 0.73 HTR2A (0.37) CA1CA2MEN1KMT2ACYP1A2
SCHEMBL10227709 0.71 CCNA2 (0.40) CA1CA2MEN1KMT2ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118206566-A Hydroxypyridooxazepine as NRF2 activator 葛兰素史密斯克莱知识产权发展有限公司 2024-06-18 CN disclosed
CN-113474349-B Hydroxypyridooxazepine as NRF2 activator 葛兰素史密斯克莱知识产权发展有限公司 2024-03-01 CN disclosed