SCHEMBL29207693

SCHEMBL29207693

C[C@H](N)C(=O)Nc1sc2c(c1C(=O)c1c(F)cccc1F)CCC1(CC2)OC=CO1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.40
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
KDM4E B2RXH2 1/20 0.40
GAA P10253 1/20 0.40
HPGD P15428 1/20 0.40
HTT P42858 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
PDE4B Q07343 1/20 0.40
CNR2 P34972 7/20 0.38
CNR1 P21554 5/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
LMNA P02545 1/20 0.38
TLR2 O60603 2/20 0.35
FLT3 P36888 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29207696 1.00 MAPT (0.40) MAPTNPC1RAB9AKDM4EGAA
SCHEMBL30395427 0.91 PTPN1 (0.41) MAPTNPC1RAB9AKDM4EGAA
SCHEMBL29207661 0.89 NPC1 (0.41) MAPTNPC1RAB9AKDM4EGAA
SCHEMBL29207667 0.89 NPC1 (0.41) MAPTNPC1RAB9AKDM4EGAA
SCHEMBL30133150 0.84 MEN1 (0.54) MAPTNPC1RAB9AKDM4EGAA
SCHEMBL29207628 0.83 RAB9A (0.54) MAPTNPC1RAB9AKDM4EGAA
SCHEMBL29207766 0.83 RAB9A (0.54) MAPTNPC1RAB9AKDM4EGAA
SCHEMBL29207713 0.82 NPC1 (0.44) MAPTNPC1RAB9AKDM4EGAA
SCHEMBL30395849 0.81 PTPN1 (0.42) MAPTNPC1RAB9AKDM4EGAA
SCHEMBL29207705 0.81 RAB9A (0.42) MAPTNPC1RAB9AKDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118019745-A Cyclohepta-thieno-diazapine derivatives as positive allosteric modulators of the GABAA gamma 1 receptor 豪夫迈·罗氏有限公司 2024-05-10 CN disclosed