SCHEMBL2922410

SCHEMBL2922410

CC(C)[C@@H](C(=O)N[C@H](C#N)Cc1c(F)cc(C#N)cc1F)N(CC(F)(F)F)c1ccc(-c2ccc([C@@H](O)C(F)F)cc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CTSL P07711 16/20 0.56
CTSB P07858 14/20 0.56
CTSF Q9UBX1 14/20 0.56
CTSK P43235 6/20 0.56
CTSS P25774 4/20 0.56
CTSV O60911 3/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2921216 0.92 CTSL (0.68) CTSLCTSBCTSFCTSKCTSS
SCHEMBL2926442 0.81 CTSL (0.83) CTSLCTSBCTSFCTSKCTSS
SCHEMBL3760800 0.81 CTSL (0.83) CTSLCTSBCTSFCTSKCTSS
SCHEMBL3760797 0.81 CTSL (0.83) CTSLCTSBCTSFCTSKCTSS
SCHEMBL3036190 0.75 CTSL (0.51) CTSLCTSBCTSFCTSKCTSS
SCHEMBL3771576 0.73 CTSL (0.73) CTSLCTSBCTSFCTSKCTSS
SCHEMBL3771569 0.73 CTSL (0.73) CTSLCTSBCTSFCTSKCTSS
SCHEMBL3771579 0.73 CTSL (0.73) CTSLCTSBCTSFCTSKCTSS
SCHEMBL3767031 0.72 CTSL (1.00) CTSLCTSBCTSFCTSKCTSS
SCHEMBL3767027 0.72 CTSL (1.00) CTSLCTSBCTSFCTSKCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2225196-A1 CYSTEINE PROTEASE INHIBITORS FOR THE TREATMENT OF PARASITIC DISEASES Merck Frosst Canada Ltd. (CA) 2010-09-08 EP claimed
WO-2009067797-A1 CYSTEINE PROTEASE INHIBITORS FOR THE TREATMENT OF PARASITIC DISEASES MERCK FROSST CANADA LTD. (CA) 2009-06-04 WO claimed