SCHEMBL29226367

SCHEMBL29226367

CC(C)(C)OC(=O)N1Cc2ccc([Sn](C)(C)C)nc2C1=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 2/20 0.38
MTOR P42345 2/20 0.38
ESR2 Q92731 1/20 0.38
NR1H2 P55055 2/20 0.38
CHRM4 P08173 1/20 0.33
DRD2 P14416 1/20 0.33
HTR7 P34969 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
KDM1A O60341 1/20 0.33
MAPK1 P28482 1/20 0.33
HDAC1 Q13547 2/20 0.32
DDB1 Q16531 1/20 0.32
CRBN Q96SW2 1/20 0.32
CKS1B P61024 1/20 0.32
SKP1 P63208 1/20 0.32
SKP2 Q13309 1/20 0.32
DHODH Q02127 1/20 0.32
HDAC6 Q9UBN7 1/20 0.31
ELANE P08246 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21847688 0.83 PIK3CA (0.40) PIK3CAMTORESR2NR1H2MEN1
SCHEMBL29226277 0.82 PIK3CA (0.39) PIK3CAMTORESR2NR1H2CHRM4
SCHEMBL21847679 0.82 ESR2 (0.40) PIK3CAMTORESR2NR1H2CHRM4
SCHEMBL21847682 0.80 PIK3CA (0.38) PIK3CAMTORESR2NR1H2CHRM4
SCHEMBL23554273 0.79 NR1H2 (0.41) PIK3CAMTORESR2NR1H2CHRM4
SCHEMBL21847689 0.76 PIK3CA (0.36) PIK3CAMTORESR2NR1H2MEN1
SCHEMBL21847643 0.75 MAPK1 (0.45) PIK3CAMTORMAPK1DDB1CRBN
SCHEMBL23771943 0.69 KDM4E (0.51) PIK3CAMTORMEN1KMT2AKDM1A
SCHEMBL29814717 0.69 KDM4E (0.51) PIK3CAMTORMEN1KMT2AKDM1A
SCHEMBL21461289 0.69 ESR2 (0.53) PIK3CAMTORESR2NR1H2CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117658987-A Compounds as PLK1 inhibitors, and preparation method and application thereof 上海深势唯思科技有限责任公司 2024-03-08 CN disclosed