SCHEMBL29250063

SCHEMBL29250063

CN(C)c1ccc(Nc2nccc(-c3ccc(=O)n(C)c3)n2)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 1/20 0.62
IKBKB O14920 4/20 0.52
CDK2 P24941 3/20 0.51
CDK4 P11802 2/20 0.51
CCNE1 P24864 2/20 0.51
AURKA O14965 1/20 0.51
CDK1 P06493 1/20 0.51
CDK7 P50613 1/20 0.51
CDK9 P50750 1/20 0.51
AURKB Q96GD4 1/20 0.51
CAMK2D Q13557 2/20 0.46
SCN9A Q15858 1/20 0.46
ABL1 P00519 1/20 0.45
BCR P11274 1/20 0.45
JAK2 O60674 3/20 0.45
JAK3 P52333 1/20 0.45
PIK3CA P42336 3/20 0.43
PIK3CB P42338 3/20 0.43
PIK3CG P48736 3/20 0.43
MAPK8 P45983 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30237272 1.00 DYRK1A (0.62) DYRK1AIKBKBCDK2CDK4CCNE1
SCHEMBL29250285 0.86 CDK2 (0.56) DYRK1AIKBKBCDK2CDK4CCNE1
SCHEMBL30236813 0.86 CDK2 (0.56) DYRK1AIKBKBCDK2CDK4CCNE1
SCHEMBL30237443 0.83 CDK2 (0.50) DYRK1AIKBKBCDK2CDK4CCNE1
SCHEMBL29250121 0.83 CDK2 (0.50) DYRK1AIKBKBCDK2CDK4CCNE1
SCHEMBL30236998 0.82 IKBKB (0.46) DYRK1AIKBKBCDK2CDK4CCNE1
SCHEMBL29250039 0.82 IKBKB (0.46) DYRK1AIKBKBCDK2CDK4CCNE1
SCHEMBL30237191 0.79 CDK2 (0.49) DYRK1ACDK2CDK4CCNE1AURKA
SCHEMBL29250067 0.79 CDK2 (0.49) DYRK1ACDK2CDK4CCNE1AURKA
SCHEMBL7467187 0.77 CDK2 (0.60) IKBKBCDK2CDK4CCNE1AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115703760-B 2, 4-Disubstituted pyrimidine cyclin dependent kinase enzyme inhibitor and preparation method and application thereof 山东大学 2024-05-31 CN disclosed
CN-115703760-A 2,4-disubstituted pyrimidines cyclin dependent kinase inhibitor and preparation method and application thereof 山东大学 2023-02-17 CN disclosed