SCHEMBL30237191

SCHEMBL30237191

CN(C)c1ccc(Nc2ncc(F)c(-c3ccc(=O)n(C)c3)n2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 10/20 0.49
CCNE1 P24864 6/20 0.49
CDK1 P06493 5/20 0.49
CCNB1 P14635 5/20 0.49
CCNT1 O60563 5/20 0.49
CDK9 P50750 5/20 0.49
CCNE2 O96020 4/20 0.49
CCNB2 O95067 3/20 0.49
CDK5 Q00535 3/20 0.49
CDK5R1 Q15078 3/20 0.49
CCNB3 Q8WWL7 3/20 0.49
JAK2 O60674 2/20 0.43
CCNA2 P20248 2/20 0.43
AXL P30530 1/20 0.43
CCNA1 P78396 1/20 0.43
CDK4 P11802 4/20 0.42
CCND3 P30281 2/20 0.42
CDK6 Q00534 1/20 0.42
DYRK1A Q13627 1/20 0.41
IGF1R P08069 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29250067 1.00 CDK2 (0.49) CDK2CCNE1CDK1CCNB1CCNT1
SCHEMBL30237260 0.87 CDK2 (0.46) CDK2CCNE1CDK1CCNB1CCNT1
SCHEMBL29250163 0.87 CDK2 (0.46) CDK2CCNE1CDK1CCNB1CCNT1
SCHEMBL30237057 0.84 CDK2 (0.43) CDK2CCNE1CDK1CCNB1CCNT1
SCHEMBL29250118 0.84 CDK2 (0.43) CDK2CCNE1CDK1CCNB1CCNT1
SCHEMBL30237004 0.83 CDK2 (0.44) CDK2CCNE1CDK1CCNB1CCNT1
SCHEMBL29250102 0.83 CDK2 (0.44) CDK2CCNE1CDK1CCNB1CCNT1
SCHEMBL30237272 0.79 DYRK1A (0.62) CDK2CCNE1CDK1CDK9JAK2
SCHEMBL29250063 0.79 DYRK1A (0.62) CDK2CCNE1CDK1CDK9JAK2
SCHEMBL654899 0.72 AURKA (0.69) CDK2CDK1CDK5JAK2AXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115703760-B 2, 4-Disubstituted pyrimidine cyclin dependent kinase enzyme inhibitor and preparation method and application thereof 山东大学 2024-05-31 CN disclosed
CN-115703760-A 2,4-disubstituted pyrimidines cyclin dependent kinase inhibitor and preparation method and application thereof 山东大学 2023-02-17 CN disclosed