SCHEMBL2926162

SCHEMBL2926162

O=S(=O)(Nc1cccc2nc(NC3CCc4ccccc43)ccc12)c1cc(F)cc(F)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN1A P35498 4/20 0.41
SCN5A Q14524 4/20 0.41
SCN8A Q9UQD0 4/20 0.41
PFKFB3 Q16875 1/20 0.37
GBA1 P04062 1/20 0.37
MAPT P10636 2/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
KMT2A Q03164 1/20 0.36
BRS3 P32247 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
KDM4E B2RXH2 2/20 0.36
LMNA P02545 2/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
FADS1 O60427 1/20 0.36
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1615546 1.00 SCN1A (0.41) SCN1ASCN5ASCN8APFKFB3GBA1
SCHEMBL1616498 0.95 PFKFB3 (0.44) SCN1ASCN5ASCN8APFKFB3GBA1
SCHEMBL1616265 0.93 SCN1A (0.41) SCN1ASCN5ASCN8APFKFB3GBA1
SCHEMBL2919481 0.93 SCN1A (0.41) SCN1ASCN5ASCN8APFKFB3GBA1
SCHEMBL1616346 0.92 MEN1 (0.46) SCN1ASCN5ASCN8APFKFB3GBA1
SCHEMBL1615576 0.86 CA1 (0.38) PFKFB3MAPTMEN1ALDH1A1KMT2A
SCHEMBL1615372 0.85 PKM (0.39) MAPTALDH1A1KMT2AKDM4EGAA
SCHEMBL1616597 0.84 MAP2K4 (0.38) PFKFB3MAPTMEN1ALDH1A1KMT2A
SCHEMBL1615436 0.83 MAPT (0.36) MAPTMEN1ALDH1A1KMT2AGAA
SCHEMBL1616691 0.83 PFKFB3 (0.39) SCN1ASCN5ASCN8APFKFB3GBA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2099763-B1 2-AMINOQUINOLINES AS 5-HT(5A) RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-08-11 EP disclosed