SCHEMBL2926867

SCHEMBL2926867

CCOC(=O)c1ccc(Nc2ncc(F)c(-c3cnc(C)n3C(C)C)n2)cc1F

nearest known ligand 0.77

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 11/20 0.77
CDK2 P24941 15/20 0.75
CDK1 P06493 6/20 0.66
CDK4 P11802 1/20 0.59
CDKL1 Q00532 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1447285 0.88 CDK2 (0.76) KCNH2CDK2CDK1
SCHEMBL30828131 0.88 CDK2 (0.76) KCNH2CDK2CDK1
SCHEMBL2924704 0.87 KCNH2 (0.82) KCNH2CDK2CDK1CDK4CDKL1
SCHEMBL4250988 0.86 CDK2 (0.65) KCNH2CDK2CDK1CDK4CDKL1
Lithium Ion SCHEMBL2924705 0.86 KCNH2 (0.81) KCNH2CDK2CDK1CDK4CDKL1
SCHEMBL4516321 0.85 CDK2 (1.00) KCNH2CDK2CDK1CDK4CDKL1
SCHEMBL4864875 0.85 KCNH2 (0.73) KCNH2CDK2CDK1CDK4CDKL1
SCHEMBL2924335 0.84 CDK2 (0.81) KCNH2CDK2CDK1CDK4CDKL1
SCHEMBL2925264 0.83 CDK2 (1.00) KCNH2CDK2CDK1CDK4CDKL1
SCHEMBL1447655 0.82 CDK2 (0.80) KCNH2CDK2CDK1CDK4CDKL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2044058-B1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2010-09-29 EP disclosed
US-20100240686-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2010-09-23 US disclosed
EP-2044058-A1 CHEMICAL COMPOUNDS AstraZeneca AB (SE) 2009-04-08 EP disclosed
WO-2007148070-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2007-12-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100240686-A1 CHEMICAL COMPOUNDS CCNI, CDKN1A, CCNB1 KCNH2 2925/4885CDK2 11/4885CDK1 12/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.