SCHEMBL2926940

SCHEMBL2926940

COc1ccc(S(=O)(=O)N2[C@@H](OC(=O)O)C[C@@H]3CCN(C(=O)OCc4ccccc4)C[C@@H]32)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP9 P14780 4/20 0.56
MMP2 P08253 2/20 0.56
MMP12 P39900 1/20 0.56
MMP1 P03956 3/20 0.56
MMP3 P08254 3/20 0.56
MMP7 P09237 3/20 0.56
MMP13 P45452 2/20 0.56
MMP8 P22894 1/20 0.54
CHRM2 P08172 1/20 0.48
CHRM1 P11229 1/20 0.48
PKM P14618 2/20 0.45
ALDH1A1 P00352 1/20 0.45
HTT P42858 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
CHRM5 P08912 1/20 0.44
F13A1 P00488 3/20 0.43
TGM2 P21980 3/20 0.43
TGM1 P22735 3/20 0.43
GRIN2B Q13224 1/20 0.43
MEN1 O00255 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1656829 0.88 MMP9 (0.64) MMP9MMP2MMP12MMP1MMP3
SCHEMBL5546856 0.88 MMP9 (0.64) MMP9MMP2MMP12MMP1MMP3
SCHEMBL2927761 0.85 MMP9 (0.53) MMP9MMP2MMP12MMP1MMP3
SCHEMBL1655593 0.85 MMP9 (0.77) MMP9MMP2MMP12MMP1MMP3
SCHEMBL1655818 0.85 MMP9 (0.60) MMP9MMP2MMP12MMP1MMP3
SCHEMBL2928187 0.85 MMP9 (0.52) MMP9MMP2MMP12MMP1MMP3
SCHEMBL2927874 0.84 MMP9 (0.65) MMP9MMP2MMP12MMP1MMP3
SCHEMBL1656110 0.84 MMP9 (0.65) MMP9MMP2MMP12MMP1MMP3
SCHEMBL2927673 0.83 MMP9 (0.54) MMP9MMP2MMP12MMP1MMP3
SCHEMBL2927653 0.76 MMP9 (0.68) MMP9MMP2MMP12MMP1MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1768979-B1 OCTAHYDROPYRROLO[2, 3, C]PYRIDINE DERIVATIVES AND PHARMACEUTICAL USE THEREOF MERCK SERONO SA (CH) 2010-09-29 EP claimed