SCHEMBL2927604

SCHEMBL2927604

Cc1ccc(CNc2ccc3c(N[C@H]4CCS(=O)(=O)c5ccccc54)cccc3n2)o1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
TSHR P16473 1/20 0.33
NPY5R Q15761 1/20 0.32
HRH4 Q9H3N8 1/20 0.31
MAPK1 P28482 1/20 0.31
P2RX7 Q99572 2/20 0.31
ADRA1D P25100 3/20 0.31
HTT P42858 2/20 0.31
TRPC5 Q9UL62 1/20 0.30
MEN1 O00255 2/20 0.30
KMT2A Q03164 2/20 0.30
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
GAA P10253 1/20 0.30
MAPT P10636 1/20 0.30
LMNA P02545 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
IGF1R P08069 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2908838 1.00 NPC1 (0.36) NPC1RAB9ATSHRNPY5RHRH4
SCHEMBL2909652 0.83 NPC1 (0.39) NPC1RAB9ATSHRNPY5RHTT
SCHEMBL2901511 0.82 NPC1 (0.38) NPC1RAB9ATSHRNPY5RHRH4
SCHEMBL2907255 0.75 KMT2A (0.31) MAPK1KMT2AALDH1A1LMNA
SCHEMBL2906805 0.74 NPC1 (0.46) NPC1RAB9ATSHRNPY5RHRH4
SCHEMBL2245184 0.74 NPC1 (0.39) NPC1RAB9ATSHRNPY5RHRH4
SCHEMBL2908410 0.73 NPC1 (0.46) NPC1RAB9ATSHRNPY5RMAPK1
SCHEMBL2245273 0.71 BRD4 (0.41) NPC1RAB9ATSHRNPY5RHTT
SCHEMBL2907371 0.71 MAPT (0.45) NPC1RAB9ATSHRHTTMEN1
SCHEMBL2907292 0.71 NPC1 (0.42) NPC1RAB9ATSHRNPY5RMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7825253-B2 2-aminoquinoline derivatives HOFFMANN-LA ROCHE INC. (US) 2010-11-02 US claimed
EP-2076495-B1 QUINOLINE DERIVATIVES WITH 5-HT-BINDING PROPERTIES HOFFMANN LA ROCHE (CH) 2010-08-18 EP claimed
US-7825253-B2 2-aminoquinoline derivatives HOFFMANN-LA ROCHE INC. (US) 2010-11-02 US disclosed