SCHEMBL29280456

SCHEMBL29280456

COC(=O)c1cc(CCl)nc2ccccc12

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.72
PLA2G2A P14555 5/20 0.57
MEN1 O00255 6/20 0.54
KMT2A Q03164 6/20 0.54
ALDH1A1 P00352 7/20 0.53
HPGD P15428 3/20 0.53
POLB P06746 2/20 0.53
PKM P14618 2/20 0.53
MAPK1 P28482 2/20 0.53
TDP1 Q9NUW8 2/20 0.53
PLIN1 O60240 1/20 0.53
LMNA P02545 1/20 0.53
GLA P06280 1/20 0.53
PLIN5 Q00G26 1/20 0.53
MCL1 Q07820 1/20 0.53
ABHD5 Q8WTS1 1/20 0.53
DHODH Q02127 1/20 0.53
MAPT P10636 4/20 0.52
USP2 O75604 1/20 0.52
TP53 P04637 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30365659 0.84 KDM4E (1.00) KDM4EMEN1KMT2AALDH1A1HPGD
SCHEMBL1900613 0.84 KDM4E (1.00) KDM4EMEN1KMT2AALDH1A1HPGD
SCHEMBL1228082 0.81 KDM4E (0.58) KDM4EPLA2G2AMEN1KMT2AALDH1A1
SCHEMBL14518623 0.80 MEN1 (0.72) KDM4EPLA2G2AMEN1KMT2AALDH1A1
SCHEMBL30604170 0.80 PLA2G2A (0.61) KDM4EPLA2G2AMEN1KMT2AALDH1A1
SCHEMBL30604167 0.80 PLA2G2A (0.61) KDM4EPLA2G2AMEN1KMT2AALDH1A1
SCHEMBL72379 0.79 KDM4E (0.70) KDM4EPLA2G2AMEN1KMT2AALDH1A1
SCHEMBL12903095 0.79 KDM4E (0.70) KDM4EMEN1KMT2AALDH1A1HPGD
SCHEMBL31295407 0.79 KDM4E (0.70) KDM4EMEN1KMT2AALDH1A1HPGD
SCHEMBL663977 0.79 KDM4E (0.70) KDM4EPLA2G2AMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117751107-A Organic pyridine-pyrazole compounds and uses thereof 博善人工智能剑桥有限公司 2024-03-22 CN disclosed