SCHEMBL29280765

SCHEMBL29280765

COC[C@H]1C=C(OS(=O)(=O)C(F)(F)F)CN1C(=O)OC(C)(C)C

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 2/20 0.34
NR1H2 P55055 9/20 0.33
NR1H3 Q13133 9/20 0.33
HCRTR2 O43614 1/20 0.32
HSD11B1 P28845 1/20 0.32
STS P08842 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12300565 0.91 PTPN1 (0.33) PTPN1NR1H2NR1H3HCRTR2HSD11B1
SCHEMBL19078443 0.87 ALDH1A1 (0.32) PTPN1NR1H2NR1H3HCRTR2HSD11B1
SCHEMBL29280764 0.83 SMYD2 (0.35) PTPN1NR1H2NR1H3HCRTR2STS
SCHEMBL25366552 0.83 SMYD2 (0.35) PTPN1NR1H2NR1H3HCRTR2STS
SCHEMBL12248021 0.82 NR1H2 (0.35) PTPN1NR1H2NR1H3HSD11B1STS
SCHEMBL15388623 0.81 NR1H2 (0.34) PTPN1NR1H2NR1H3HSD11B1STS
SCHEMBL14857161 0.81 NR1H2 (0.34) PTPN1NR1H2NR1H3HSD11B1STS
SCHEMBL3557230 0.81 PTPN1 (0.41) PTPN1NR1H2NR1H3HSD11B1STS
SCHEMBL1662643 0.81 PTPN1 (0.41) PTPN1NR1H2NR1H3HSD11B1STS
SCHEMBL1662641 0.81 PTPN1 (0.41) PTPN1NR1H2NR1H3HSD11B1STS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4359402-B1 IMIDAZOLO INDAZOLE COMPOUNDS AS JAK INHIBITORS THERAVANCE BIOPHARMA R&D IP LLC (US) 2026-03-11 EP disclosed
US-12384761-B2 Imidazolo indazole compounds as JAK inhibitors THERAVANCE BIOPHARMA R&D IP, LLC (US) 2025-08-12 US disclosed
EP-4359402-A1 IMIDAZOLO INDAZOLE COMPOUNDS AS JAK INHIBITORS Theravance Biopharma R&D IP, LLC (US) 2024-05-01 EP disclosed
CN-117813298-A Imidazole indazole compounds as JAK inhibitors 施万生物制药研发IP有限责任公司 2024-04-02 CN disclosed
US-20240092758-A1 IMIDAZOLO INDAZOLE COMPOUNDS AS JAK INHIBITORS THERAVANCE BIOPHARMA R&D IP, LLC 2024-03-21 US disclosed
WO-2022272020-A1 IMIDAZOLO INDAZOLE COMPOUNDS AS JAK INHIBITORS THERAVANCE BIOPHARMA R&D IP, LLC (US) 2022-12-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240092758-A1 IMIDAZOLO INDAZOLE COMPOUNDS AS JAK INHIBITORS JAK1, JAK3, JAK2 PTPN1 204/4885NR1H2 2644/4885NR1H3 3165/4885
US-12384761-B2 Imidazolo indazole compounds as JAK inhibitors JAK1, JAK3, JAK2 PTPN1 204/4885NR1H2 2644/4885NR1H3 3165/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.