SCHEMBL29280877

SCHEMBL29280877

Cc1cccnc1C(=O)NCC1CCN(CC(=O)c2ccc(F)cc2)CC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.50
ALDH1A1 P00352 1/20 0.50
TSHR P16473 1/20 0.50
HTT P42858 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
LMNA P02545 3/20 0.45
HTR2A P28223 8/20 0.44
HTR2C P28335 5/20 0.44
KCNH2 Q12809 1/20 0.44
HTR1A P08908 1/20 0.44
TMEM97 Q5BJF2 1/20 0.44
GSK3B P49841 1/20 0.44
TP53 P04637 1/20 0.43
THRB P10828 1/20 0.43
GAA P10253 1/20 0.42
DRD2 P14416 2/20 0.42
HTR2B P41595 2/20 0.42
SIGMAR1 Q99720 2/20 0.42
HTR7 P34969 2/20 0.41
CACNA1G O43497 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL29280926 0.83 KDM4E (0.45) KDM4EALDH1A1TSHRHTTSMN1; SMN2
SCHEMBL30840071 0.83 MEN1 (0.55) KDM4EALDH1A1TSHRHTTSMN1; SMN2
SCHEMBL29280894 0.83 MEN1 (0.55) KDM4EALDH1A1TSHRHTTSMN1; SMN2
SCHEMBL29280918 0.83 GABRA5 (0.47) KDM4EALDH1A1TSHRHTTSMN1; SMN2
SCHEMBL29280913 0.81 CACNA1I (0.52) KDM4EALDH1A1TSHRHTTSMN1; SMN2
SCHEMBL29280878 0.80 KDM4E (0.45) KDM4EALDH1A1TSHRHTTSMN1; SMN2
SCHEMBL30843813 0.80 HTR2A (0.44) KDM4EALDH1A1TSHRHTTSMN1; SMN2
SCHEMBL29280920 0.80 HTR2A (0.44) KDM4EALDH1A1TSHRHTTSMN1; SMN2
SCHEMBL29280933 0.80 F10 (0.51) KDM4EALDH1A1TSHRHTTSMN1; SMN2
SCHEMBL29280915 0.80 HTR2A (0.61) KDM4EHTR2AHTR2CKCNH2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117820199-A Amide compound and application thereof in preparation of Sigma2 and 5HT2A inhibitors 瀚远医药有限公司 2024-04-05 CN disclosed