SCHEMBL29282135

SCHEMBL29282135

Cc1c(NC(C)C)cccc1-c1cccc2c1cnn2C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 1/20 0.41
CCR4 P51679 1/20 0.39
KAT2B Q92831 1/20 0.38
KDM1A O60341 1/20 0.37
IRAK4 Q9NWZ3 1/20 0.37
TP53 P04637 2/20 0.37
FAAH O00519 1/20 0.37
JAK2 O60674 1/20 0.36
JAK3 P52333 1/20 0.36
PTK2 Q05397 1/20 0.36
SYK P43405 1/20 0.36
PDCD1 Q15116 1/20 0.36
CD274 Q9NZQ7 1/20 0.36
BRD4 O60885 2/20 0.36
CREBBP Q92793 1/20 0.36
ABL1 P00519 1/20 0.35
CYP17A1 P05093 1/20 0.34
CYP1A2 P05177 1/20 0.34
KDM4E B2RXH2 1/20 0.34
NPC1 O15118 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8312915 0.70 CCR4 (0.55) CCR4KAT2BTP53TRPV1
SCHEMBL19945232 0.69 PDCD1 (0.52) KDRCCR4TP53FAAHJAK2
SCHEMBL29282122 0.68 KDR (0.40) KDRCCR4FAAHJAK2JAK3
SCHEMBL24312500 0.68 CCR4 (0.38) KDRCCR4TP53FAAHJAK2
SCHEMBL13707016 0.68 CCR4 (0.53) CCR4TP53TRPV1
SCHEMBL31130330 0.68 CCR4 (0.50) KDRCCR4TP53SYKTRPV1
SCHEMBL11806943 0.68 TDP1 (0.44) KDM1AKDM4ELMNATSHRHTT
SCHEMBL256207 0.67 CYP11B1 (0.43) KDRCCR4TP53CYP1A2NPC1
SCHEMBL25628273 0.67 KDM4E (0.38) KDRCCR4IRAK4FAAHJAK2
SCHEMBL15077331 0.66 CCR4 (0.39) KDRCCR4FAAHSYKCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117986241-A Biphenyl derivative, pharmaceutical composition and application thereof 武汉睿健医药科技有限公司 2024-05-07 CN disclosed