SCHEMBL29288229

SCHEMBL29288229

O=CNC1CN(Cc2ccc(OCc3cccc(Cl)c3)cc2)C1

nearest known ligand 0.65

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
S1PR5 Q9H228 5/20 0.65
S1PR1 P21453 4/20 0.65
MAOB P27338 5/20 0.52
GID4 Q8IVV7 1/20 0.50
RXRA P19793 1/20 0.48
RXRB P28702 1/20 0.48
RXRG P48443 1/20 0.48
PDGFRA P16234 1/20 0.47
HTR2A P28223 1/20 0.47
KCNH2 Q12809 1/20 0.47
SIGMAR1 Q99720 1/20 0.47
MAOA P21397 1/20 0.47
ALOX5 P09917 1/20 0.46
LTK P29376 1/20 0.45
TAOK1 Q7L7X3 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29288191 0.88 S1PR5 (0.50) S1PR5S1PR1MAOBPDGFRAHTR2A
SCHEMBL29288219 0.87 HRH3 (0.52) S1PR5S1PR1MAOBHTR2AKCNH2
SCHEMBL29288202 0.81 HRH3 (0.53) S1PR5S1PR1MAOBRXRARXRB
SCHEMBL3042052 0.79 S1PR5 (1.00) S1PR5S1PR1MAOBRXRARXRB
SCHEMBL23004599 0.79 MAOB (0.53) S1PR5S1PR1MAOBGID4RXRA
SCHEMBL29288173 0.78 S1PR5 (0.81) S1PR5S1PR1MAOBRXRARXRB
SCHEMBL3044721 0.76 MAOB (0.64) S1PR5S1PR1MAOBRXRARXRB
SCHEMBL21347483 0.76 HRH3 (0.68) S1PR5S1PR1MAOBRXRARXRB
SCHEMBL28115794 0.75 MAOB (0.69) S1PR5S1PR1MAOBGID4RXRA
SCHEMBL3423658 0.72 MAOB (0.65) MAOBGID4RXRARXRBRXRG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108912029-B Nitrogen-containing heterocyclic amide derivative and use thereof 广东东阳光药业有限公司 2021-10-01 CN disclosed