SCHEMBL29288202

SCHEMBL29288202

O=CNC1CN(Cc2ccc(OCc3ccc(Br)cc3)cc2)C1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.53
S1PR5 Q9H228 3/20 0.49
APP P05067 1/20 0.44
FAAH O00519 1/20 0.44
RXRA P19793 1/20 0.44
RXRB P28702 1/20 0.44
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA7 P43166 1/20 0.43
CA9 Q16790 1/20 0.43
MAOB P27338 1/20 0.43
S1PR1 P21453 1/20 0.43
HTR2A P28223 1/20 0.43
KCNH2 Q12809 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
UTS2R Q9UKP6 2/20 0.42
FFAR1 O14842 1/20 0.42
FFAR4 Q5NUL3 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29288219 0.89 HRH3 (0.52) HRH3S1PR5APPFAAHMAOB
SCHEMBL29288191 0.87 S1PR5 (0.50) S1PR5FAAHCA12CA9MAOB
SCHEMBL29288229 0.81 S1PR5 (0.65) S1PR5RXRARXRBMAOBS1PR1
SCHEMBL3041024 0.77 S1PR5 (0.81) HRH3S1PR5RXRARXRBS1PR1
SCHEMBL29288192 0.76 MAOB (0.66) HRH3S1PR5RXRARXRBMAOB
SCHEMBL4591941 0.74 SIGMAR1 (0.56) SIGMAR1
SCHEMBL6057451 0.74 HRH3 (0.82) HRH3
SCHEMBL3038005 0.74 HRH3 (0.77) HRH3
SCHEMBL19946503 0.71 APP (0.56) APPRXRARXRBCA12CA1
SCHEMBL2399080 0.71 APP (0.80) APPRXRARXRBCA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108912029-B Nitrogen-containing heterocyclic amide derivative and use thereof 广东东阳光药业有限公司 2021-10-01 CN disclosed