SCHEMBL2929104

SCHEMBL2929104

N#Cc1cncc(C=Cc2ccccn2)c1Nc1ccc2[nH]ccc2c1

nearest known ligand 0.76

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PRKCQ Q04759 20/20 0.76
PRKCD Q05655 15/20 0.76
LYN P07948 2/20 0.51
PRKCH P24723 2/20 0.51
PRKCE Q02156 2/20 0.51
PRKCB P05771 1/20 0.44
LCK P06239 1/20 0.44
SRC P12931 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31061266 0.87 PRKCQ (1.00) PRKCQPRKCDLYNPRKCHPRKCE
SCHEMBL2935239 0.87 PRKCQ (1.00) PRKCQPRKCDLYNPRKCHPRKCE
SCHEMBL2931620 0.80 PRKCQ (0.78) PRKCQPRKCDLYNPRKCHPRKCE
SCHEMBL2936308 0.80 PRKCQ (1.00) PRKCQPRKCDLYNPRKCHPRKCE
SCHEMBL2935272 0.80 PRKCQ (1.00) PRKCQPRKCDLYNPRKCHPRKCE
SCHEMBL2980440 0.77 PRKCQ (0.70) PRKCQPRKCDLYNPRKCHPRKCE
SCHEMBL2934690 0.77 PRKCQ (0.73) PRKCQPRKCDLYNPRKCHPRKCE
SCHEMBL2934688 0.77 PRKCQ (0.73) PRKCQPRKCDLYNPRKCHPRKCE
SCHEMBL2930136 0.76 PRKCQ (0.64) PRKCQPRKCDLYNPRKCHPRKCE
SCHEMBL2985327 0.75 PRKCQ (0.67) PRKCQPRKCDLYNPRKCHPRKCE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2229377-A1 5-ALKYL/ALKENYL-3-CYANOPYRIDINES AS KINASE INHIBITORS Wyeth LLC (US) 2010-09-22 EP claimed
WO-2009076602-A1 5-ALKYL/ALKENYL-3-CYANOPYRIDINES AS KINASE INHIBITORS WYETH (US) 2009-06-18 WO claimed
EP-2229377-A1 5-ALKYL/ALKENYL-3-CYANOPYRIDINES AS KINASE INHIBITORS Wyeth LLC (US) 2010-09-22 EP disclosed
WO-2009076602-A1 5-ALKYL/ALKENYL-3-CYANOPYRIDINES AS KINASE INHIBITORS WYETH (US) 2009-06-18 WO disclosed