SCHEMBL2929944

SCHEMBL2929944

Cc1cccc(-c2ccc(C)cc2C(=O)N2C[C@H]3C[C@H]3[C@H]2CN)c1

nearest known ligand 0.40

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 16/20 0.39
HCRTR2 O43614 15/20 0.39
CYP46A1 Q9Y6A2 2/20 0.36
CHRM1 P11229 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2928731 0.93 CYP46A1 (0.42) HCRTR1HCRTR2CYP46A1
SCHEMBL2929614 0.92 CHRM1 (0.46) HCRTR1HCRTR2CHRM1
SCHEMBL2955880 0.92 HCRTR2 (0.43) HCRTR1HCRTR2
SCHEMBL2926961 0.92 MEN1 (0.43) HCRTR1HCRTR2
SCHEMBL3414068 0.92 MEN1 (0.43) HCRTR1HCRTR2
SCHEMBL2924875 0.92 HCRTR2 (0.37) HCRTR1HCRTR2CYP46A1CHRM1
SCHEMBL2931530 0.90 HCRTR1 (0.46) HCRTR1HCRTR2
SCHEMBL2927516 0.90 CYP46A1 (0.40) HCRTR1HCRTR2CYP46A1
SCHEMBL2926254 0.86 HCRTR2 (0.40) HCRTR1HCRTR2
SCHEMBL2448034 0.86 MEN1 (0.41) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079690-B1 3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2010-09-15 EP disclosed