SCHEMBL29313754

SCHEMBL29313754

CN(C(=O)Oc1c(-n2ccn(CCN3CCNCC3)c2=O)cc(C(F)(F)F)cc1C(F)(F)F)c1ccc(F)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLQ O75417 2/20 0.37
SIGMAR1 Q99720 1/20 0.35
TACR1 P25103 6/20 0.34
MLNR O43193 2/20 0.33
SLC6A4 P31645 3/20 0.33
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
HTR1A P08908 2/20 0.31
DRD2 P14416 2/20 0.31
DRD1 P21728 2/20 0.31
DRD4 P21917 2/20 0.31
DRD5 P21918 2/20 0.31
SLC6A2 P23975 2/20 0.31
HTR1D P28221 2/20 0.31
HTR2A P28223 2/20 0.31
HTR2C P28335 2/20 0.31
HTR7 P34969 2/20 0.31
OPRM1 P35372 2/20 0.31
DRD3 P35462 2/20 0.31
OPRD1 P41143 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29313794 0.92 POLQ (0.37) POLQSIGMAR1SLC6A4MEN1KMT2A
SCHEMBL29313751 0.85 POLQ (0.39) POLQTACR1
SCHEMBL29313744 0.84 POLQ (0.38) POLQTACR1SLC6A4
SCHEMBL29313752 0.83 POLQ (0.38) POLQTACR1
SCHEMBL29313792 0.83 SLC6A2 (0.35) POLQTACR1SLC6A4SLC6A2SLC6A3
SCHEMBL29313795 0.83 POLQ (0.38) POLQ
SCHEMBL29313749 0.83 POLQ (0.38) POLQTACR1
SCHEMBL29313753 0.82 POLQ (0.37) POLQ
SCHEMBL29313799 0.82 POLQ (0.37) POLQ
SCHEMBL29313703 0.82 TACR1 (0.39) POLQTACR1SLC6A4SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024147972-A2 DNA POLYMERASE THETA INHIBITORS CONTAINING NON-SATURATED 5-MEMBERED HETEROCYCLIC RINGS AND USE THEREOF THOMAS JEFFERSON UNIVERSITY (US) 2024-07-11 WO disclosed