SCHEMBL29313802

SCHEMBL29313802

CN(C(=O)Oc1c(-n2ccn(CC(O)CN3CCC(F)C3)c2=O)cc(C(F)(F)F)cc1C(F)(F)F)c1ccc(F)cc1

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
POLQ O75417 2/20 0.34
CCR2 P41597 1/20 0.33
CYP2D6 P10635 3/20 0.32
KMT2A Q03164 1/20 0.32
TAAR1 Q96RJ0 1/20 0.32
DPP4 P27487 2/20 0.31
KCNH2 Q12809 1/20 0.31
DPP7 Q9UHL4 1/20 0.31
TRPA1 O75762 1/20 0.30
FPR2 P25090 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29313803 0.87 POLQ (0.34) POLQ
SCHEMBL29313704 0.87 POLQ (0.39) POLQ
SCHEMBL29313749 0.81 POLQ (0.38) POLQ
SCHEMBL29313794 0.80 POLQ (0.37) POLQCYP2D6KMT2AKCNH2
SCHEMBL29313698 0.80 POLQ (0.37) POLQ
SCHEMBL29313701 0.80 POLQ (0.37) POLQ
SCHEMBL29313754 0.80 POLQ (0.37) POLQKMT2A
SCHEMBL29313744 0.79 POLQ (0.38) POLQKCNH2
SCHEMBL29313708 0.79 POLQ (0.38) POLQ
SCHEMBL29313751 0.78 POLQ (0.39) POLQ

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024147972-A2 DNA POLYMERASE THETA INHIBITORS CONTAINING NON-SATURATED 5-MEMBERED HETEROCYCLIC RINGS AND USE THEREOF THOMAS JEFFERSON UNIVERSITY (US) 2024-07-11 WO disclosed