SCHEMBL2931685

SCHEMBL2931685

O=C(O)Nc1ccc(Oc2ccnc3ncc(=O)[nH]c23)cc1

nearest known ligand 0.63

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
BRAF P15056 19/20 0.63
AURKA O14965 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2932781 0.86 BRAF (0.69) BRAF
SCHEMBL3756201 0.85 BRAF (0.60) BRAF
SCHEMBL2928507 0.82 BRAF (0.71) BRAF
SCHEMBL9909761 0.82 BRAF (0.52) BRAF
SCHEMBL2930178 0.82 BRAF (0.63) BRAF
SCHEMBL2928516 0.79 BRAF (0.52) BRAF
SCHEMBL4457106 0.79 BRAF (0.73) BRAF
SCHEMBL3755881 0.78 BRAF (1.00) BRAF
SCHEMBL3190243 0.77 BRAF (1.00) BRAF
SCHEMBL2934959 0.77 BRAF (1.00) BRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3074395-A1 PROCESS FOR THE PREPARATION OF 8-(4-AMINOPHENOXY)-4H-PYRIDO[2,3-B]PYRAZIN-3-ONE DERIVATIVES Cancer Research Technology Ltd (GB) 2016-10-05 EP disclosed
WO-2015075482-A1 PROCESS FOR THE PREPARATION OF 8-(4-AMINOPHENOXY)-4H-PYRIDO[2,3-B]PYRAZIN-3-ONE DERIVATIVES CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2015-05-28 WO disclosed
EP-2229391-A1 PYRIDO[2,3-B]PYRAZINE-8-SUBSTITUTED COMPOUNDS AND THEIR USE Cancer Research Technology Limited (GB) 2010-09-22 EP disclosed
WO-2009077766-A1 PYRIDO[2,3-B]PYRAZINE-8-SUBSTITUTED COMPOUNDS AND THEIR USE CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2009-06-25 WO disclosed