SCHEMBL29317264

SCHEMBL29317264

CCCC#CCNC(C)=O

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PAOX Q6QHF9 1/20 0.40
KDM4E B2RXH2 1/20 0.39
MAPK1 P28482 1/20 0.39
HIF1A Q16665 1/20 0.39
GRIK1 P39086 1/20 0.36
GRIK2 Q13002 1/20 0.36
TSHR P16473 1/20 0.36
EPHX2 P34913 3/20 0.35
SOST Q9BQB4 1/20 0.35
ALDH1A1 P00352 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
PTPN7 P35236 3/20 0.34
HMGCR P04035 1/20 0.34
PTGS2 P35354 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13978172 0.79
SCHEMBL10739303 0.76 KDM4E (0.43) PAOXKDM4EMAPK1HIF1ATSHR
Bicarbonate SCHEMBL165177 0.75 GRIK1 (0.47) KDM4EGRIK1GRIK2EPHX2ALDH1A1
Bicarbonate SCHEMBL15968046 0.75 GRIK1 (0.47) KDM4EGRIK1GRIK2EPHX2ALDH1A1
SCHEMBL935043 0.74
SCHEMBL85842 0.74
SCHEMBL9029974 0.72
SCHEMBL7442539 0.72
SCHEMBL26448806 0.72
SCHEMBL17188612 0.72

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024147972-A2 DNA POLYMERASE THETA INHIBITORS CONTAINING NON-SATURATED 5-MEMBERED HETEROCYCLIC RINGS AND USE THEREOF THOMAS JEFFERSON UNIVERSITY (US) 2024-07-11 WO disclosed