SCHEMBL29317265

SCHEMBL29317265

CCCC#Cc1cncn1C

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 2/20 0.41
TDP1 Q9NUW8 2/20 0.37
POLQ O75417 1/20 0.34
HSP90AA1 P07900 1/20 0.33
ATM Q13315 2/20 0.33
NMT1 P30419 1/20 0.32
CYP2D6 P10635 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32
IDO1 P14902 1/20 0.32
UBE2N P61088 1/20 0.32
FNTA P49354 1/20 0.31
FNTB P49356 1/20 0.31
PGGT1B P53609 1/20 0.31
CHRNB2 P17787 1/20 0.31
CHRNA4 P43681 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21252647 0.72
SCHEMBL3347212 0.71 TDP1 (0.40) TDP1HSP90AA1ATMNMT1IDO1
SCHEMBL12590718 0.69 TDP1 (0.38) TLR7TDP1HSP90AA1ATMNMT1
SCHEMBL18430927 0.69 TDP1 (0.38) TDP1HSP90AA1ATMNMT1IDO1
SCHEMBL12820173 0.68 TDP1 (0.44) TDP1POLQHSP90AA1ATMCYP2D6
SCHEMBL378803 0.67
SCHEMBL1570065 0.67
SCHEMBL24958879 0.63 TDP1 (0.35) TDP1HSP90AA1NMT1
SCHEMBL22535086 0.63 NMT1 (0.35) TDP1POLQHSP90AA1ATMNMT1
SCHEMBL13743863 0.63 GRM5 (0.45) TDP1HSP90AA1ATMNMT1CHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024147972-A2 DNA POLYMERASE THETA INHIBITORS CONTAINING NON-SATURATED 5-MEMBERED HETEROCYCLIC RINGS AND USE THEREOF THOMAS JEFFERSON UNIVERSITY (US) 2024-07-11 WO disclosed