SCHEMBL12820173

SCHEMBL12820173

CCCc1ccccc1C#Cc1cncn1C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.44
HSP90AA1 P07900 1/20 0.38
ATM Q13315 2/20 0.37
CYP2E1 P05181 1/20 0.37
CYP2C8 P10632 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2A6 P11509 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2B6 P20813 1/20 0.37
CYP2C19 P33261 1/20 0.37
UBE2N P61088 1/20 0.36
FGFR3 P22607 2/20 0.36
KDR P35968 2/20 0.36
BRD4 O60885 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
POLQ O75417 1/20 0.34
LCK P06239 1/20 0.33
HPGDS O60760 1/20 0.33
ABL1 P00519 1/20 0.33
DDR1 Q08345 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12461563 0.82 TDP1 (0.41) TDP1HSP90AA1ATMUBE2NL3MBTL1
SCHEMBL12304052 0.82 TDP1 (0.41) TDP1HSP90AA1ATMUBE2NBRD4
SCHEMBL12461186 0.77 TDP1 (0.46) TDP1HSP90AA1ATMUBE2NBRD4
SCHEMBL6208653 0.72 TDP1 (0.52) TDP1HSP90AA1ATMUBE2NFGFR3
SCHEMBL29317265 0.68 TLR7 (0.41) TDP1HSP90AA1ATMCYP2D6UBE2N
SCHEMBL28361384 0.68 FFAR1 (0.36) TDP1CYP2E1CYP2C8CYP2D6CYP2A6
SCHEMBL1141480 0.66 HTR1A (0.38) CYP2E1CYP2C8CYP2D6CYP2A6CYP2C9
SCHEMBL17552571 0.64 TDP1 (0.42) TDP1HSP90AA1ATMUBE2NBRD4
SCHEMBL21252647 0.63
SCHEMBL3632404 0.63 TSHR (0.46) ATML3MBTL1FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011032277-A1 QUINAZOLINONE DERIVATIVES AS VIRAL POLYMERASE INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-03-24 WO disclosed