SCHEMBL2932633

SCHEMBL2932633

COc1ccccc1/C=C/c1cncc(C#N)c1Nc1ccc2[nH]ccc2c1C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PRKCQ Q04759 20/20 1.00
PRKCD Q05655 20/20 1.00
LYN P07948 1/20 0.62
PRKCH P24723 1/20 0.62
PRKCE Q02156 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2932635 1.00 PRKCQ (1.00) PRKCQPRKCDLYNPRKCHPRKCE
SCHEMBL2935241 0.89 PRKCQ (0.79) PRKCQPRKCDLYNPRKCHPRKCE
SCHEMBL2928488 0.89 PRKCQ (0.79) PRKCQPRKCDLYNPRKCHPRKCE
SCHEMBL2935077 0.89 PRKCQ (0.82) PRKCQPRKCDLYNPRKCHPRKCE
SCHEMBL2926874 0.89 PRKCQ (0.82) PRKCQPRKCDLYNPRKCHPRKCE
SCHEMBL2929003 0.87 PRKCQ (1.00) PRKCQPRKCD
SCHEMBL2929001 0.87 PRKCQ (1.00) PRKCQPRKCD
SCHEMBL2929281 0.87 PRKCQ (1.00) PRKCQPRKCD
SCHEMBL2932372 0.86 PRKCQ (0.79) PRKCQPRKCD
SCHEMBL2932371 0.86 PRKCQ (0.79) PRKCQPRKCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2229377-A1 5-ALKYL/ALKENYL-3-CYANOPYRIDINES AS KINASE INHIBITORS Wyeth LLC (US) 2010-09-22 EP claimed
WO-2009076602-A1 5-ALKYL/ALKENYL-3-CYANOPYRIDINES AS KINASE INHIBITORS WYETH (US) 2009-06-18 WO claimed
EP-2229377-A1 5-ALKYL/ALKENYL-3-CYANOPYRIDINES AS KINASE INHIBITORS Wyeth LLC (US) 2010-09-22 EP disclosed
WO-2009076602-A1 5-ALKYL/ALKENYL-3-CYANOPYRIDINES AS KINASE INHIBITORS WYETH (US) 2009-06-18 WO disclosed