SCHEMBL29366609

SCHEMBL29366609

COC(=O)c1cc(Br)cc(C(F)F)c1C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.40
NR4A2 P43354 1/20 0.37
GAA P10253 2/20 0.37
ALDH1A1 P00352 1/20 0.37
HSD17B10 Q99714 2/20 0.36
SLC6A3 Q01959 1/20 0.36
SOS1 Q07889 1/20 0.35
MAPT P10636 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
CA12 O43570 2/20 0.34
CA1 P00915 2/20 0.34
CA2 P00918 2/20 0.34
CA7 P43166 2/20 0.34
CA9 Q16790 2/20 0.34
CA14 Q9ULX7 2/20 0.34
PDK2 Q15119 1/20 0.34
PDK4 Q16654 1/20 0.34
OPRK1 P41145 1/20 0.34
HTT P42858 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26045754 1.00 NOTUM (0.40) NOTUMNR4A2GAAALDH1A1HSD17B10
SCHEMBL21932880 0.82 SLC6A4 (0.37) GAAALDH1A1HSD17B10SLC6A3SOS1
SCHEMBL19136407 0.82 NR4A2 (0.48) NR4A2GAAALDH1A1HSD17B10SLC6A3
SCHEMBL27002383 0.81 GABRA1 (0.34) ALDH1A1HSD17B10KDM4ESMN1; SMN2
SCHEMBL29915017 0.81 GABRA1 (0.34) ALDH1A1HSD17B10KDM4ESMN1; SMN2
SCHEMBL29363398 0.80 NOTUM (0.37) NOTUMNR4A2GAAALDH1A1HSD17B10
SCHEMBL22821220 0.80 NOTUM (0.37) NOTUMNR4A2GAAALDH1A1HSD17B10
SCHEMBL29841607 0.79 TPMT (0.36) GAAALDH1A1HSD17B10SLC6A3MAPT
SCHEMBL21198962 0.78 NOTUM (0.42) NOTUMNR4A2GAAALDH1A1HSD17B10
SCHEMBL29570702 0.78 NOTUM (0.42) NOTUMNR4A2GAAALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113993591-A Novel EGFR inhibitors 豪夫迈·罗氏有限公司 2022-01-28 CN disclosed