SCHEMBL2936809

SCHEMBL2936809

Nc1cc(C2CCCN(c3nc(-c4ccc(Cl)cc4Cl)nn4cnnc34)C2)c([N+](=O)[O-])c(N)n1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.33
LMNA P02545 5/20 0.33
NPSR1 Q6W5P4 3/20 0.33
ALDH1A1 P00352 3/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
HSP90AA1 P07900 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
GSK3B P49841 2/20 0.32
HTT P42858 2/20 0.32
GAA P10253 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
ADORA2A P29274 1/20 0.31
ADORA2B P29275 1/20 0.31
RPS6KB1 P23443 2/20 0.31
PROKR1 Q8TCW9 2/20 0.30
HRH4 Q9H3N8 1/20 0.30
HRH3 Q9Y5N1 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2C9 P11712 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4280024 0.99 MAPT (0.33) MAPTLMNANPSR1ALDH1A1SMN1; SMN2
SCHEMBL13658210 0.79 GSK3B (0.39) MAPTLMNANPSR1ALDH1A1L3MBTL1
Hydrochloric Acid SCHEMBL4280021 0.74
SCHEMBL3615413 0.73 LMNA (0.36) MAPTLMNANPSR1ALDH1A1SMN1; SMN2
SCHEMBL2930956 0.71 GSK3B (0.43) GSK3BHRH4CYP3A4
SCHEMBL2933462 0.70 GSK3B (0.41) GSK3B
SCHEMBL2935250 0.67 JAK3 (0.42) GSK3B
SCHEMBL2935280 0.65 MAPT (0.44) MAPTLMNAALDH1A1HTT
SCHEMBL2419126 0.56 SSTR5 (0.47) ALDH1A1SMN1; SMN2
SCHEMBL404520 0.55 HRH4 (0.71) MAPTALDH1A1HTTHRH4HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2229392-A1 TRIAZOLOTRIAZINES AND TRIAZOLOPYRAZINES AND THEIR USE AS GSK3BETA INHIBITORS Bayer Schering Pharma Aktiengesellschaft (DE) 2010-09-22 EP disclosed
WO-2009074259-A1 TRIAZOLOTRIAZINES AND TRIAZOLOPYRAZINES AND THE USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2009-06-18 WO disclosed