SCHEMBL29368403

SCHEMBL29368403

FC(F)(F)c1ccc(Cn2c(CN3CCCC3)nc3ccccc32)cc1

nearest known ligand 0.98

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.74
CYP2D6 P10635 2/20 0.74
CYP2C9 P11712 2/20 0.74
CYP2C19 P33261 2/20 0.74
MEN1 O00255 2/20 0.74
KMT2A Q03164 2/20 0.74
ALDH1A1 P00352 1/20 0.74
HIF1A Q16665 2/20 0.73
TDP1 Q9NUW8 2/20 0.73
NR1I2 O75469 1/20 0.73
ABCB11 O95342 1/20 0.73
LMNA P02545 1/20 0.73
ESR1 P03372 1/20 0.73
PGR P06401 1/20 0.73
CYP3A4 P08684 1/20 0.73
PKM P14618 1/20 0.73
TSHR P16473 1/20 0.73
ADRA2B P18089 1/20 0.73
HTR2A P28223 1/20 0.73
ADRA1A P35348 1/20 0.73

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21083242 1.00 CYP1A2 (0.74) CYP1A2CYP2D6CYP2C9CYP2C19MEN1
Clemizole SCHEMBL29938 0.85 HIF1A (1.00) CYP1A2CYP2D6CYP2C9CYP2C19MEN1
SCHEMBL13508637 0.85 CYP1A2 (0.82) CYP1A2CYP2D6CYP2C9CYP2C19MEN1
Clemizole SCHEMBL29403196 0.85 HIF1A (1.00) CYP1A2CYP2D6CYP2C9CYP2C19MEN1
SCHEMBL15568337 0.84 CYP1A2 (0.97) CYP1A2CYP2D6CYP2C9CYP2C19MEN1
SCHEMBL13144806 0.84 CYP1A2 (0.80) CYP1A2CYP2D6CYP2C9CYP2C19MEN1
Clemizole SCHEMBL19976072 0.84 HIF1A (0.97) CYP1A2CYP2D6CYP2C9CYP2C19MEN1
Clemizole SCHEMBL31707402 0.84 HIF1A (1.00) CYP1A2CYP2D6CYP2C9CYP2C19MEN1
Clemizole SCHEMBL19976068 0.84 HIF1A (0.97) CYP1A2CYP2D6CYP2C9CYP2C19MEN1
Clemizole SCHEMBL210095 0.84 HIF1A (1.00) CYP1A2CYP2D6CYP2C9CYP2C19MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3976187-A1 METHODS AND COMPOSITIONS FOR TREATING EPILEPSY The Regents of the University of California (US) 2022-04-06 EP disclosed
CN-114007692-A Methods and compositions for treating epilepsy 加利福尼亚大学董事会 2022-02-01 CN disclosed