Xenytropium

Xenytropium

SCHEMBL29371652

C[N+]1(Cc2ccc(-c3ccccc3)cc2)C2CCC1CC(OC(=O)C(CO)c1ccccc1)C2.[Br-]

nearest known ligand 0.71

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHKACHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGHRH2OPRM1

The experimentally established mechanism targets of Xenytropium. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 known ✓ P08172 8/20 0.69
CHRM5 known ✓ P08912 6/20 0.66
CHRM1 known ✓ P11229 6/20 0.66
CHRM3 known ✓ P20309 5/20 0.66
CHRM4 known ✓ P08173 4/20 0.66
BLM P54132 4/20 0.71
PABPC1 P11940 1/20 0.68
CYP2C19 P33261 1/20 0.67
MEN1 O00255 3/20 0.66
KMT2A Q03164 3/20 0.66
SMN1; SMN2 Q16637 2/20 0.66
TSHR P16473 2/20 0.66
CYP3A4 P08684 1/20 0.57
CYP2C9 P11712 1/20 0.57
HIF1A Q16665 1/20 0.57
HSD17B10 Q99714 1/20 0.57
KDM4E B2RXH2 1/20 0.55
LMNA P02545 1/20 0.55
POLB P06746 1/20 0.55
ADRA2C P18825 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Xenytropium SCHEMBL24707 1.00 BLM (0.71) BLMCHRM2PABPC1CYP2C19CHRM5
Xenytropium SCHEMBL30428452 0.99 CHRM2 (0.71) BLMCHRM2PABPC1CYP2C19CHRM5
Xenytropium SCHEMBL29361010 0.99 CHRM2 (0.71) BLMCHRM2PABPC1CYP2C19CHRM5
Bromide SCHEMBL29840597 0.94 BLM (0.77) BLMCHRM2PABPC1CYP2C19CHRM5
Butropium SCHEMBL1650524 0.87 BLM (0.64) BLMCHRM2PABPC1CYP2C19CHRM5
Butropium SCHEMBL26023 0.87 BLM (0.64) BLMCHRM2PABPC1CYP2C19CHRM5
Butropium SCHEMBL30185784 0.87 BLM (0.64) BLMCHRM2PABPC1CYP2C19CHRM5
Butropium SCHEMBL11561521 0.87 BLM (0.64) BLMCHRM2PABPC1CYP2C19CHRM5
Fentonium SCHEMBL30186606 0.86 BLM (0.69) BLMCHRM2PABPC1CYP2C19CHRM5
Fentonium SCHEMBL24583 0.86 BLM (0.69) BLMCHRM2PABPC1CYP2C19CHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115034225-A Word processing method and device applied to medical field, electronic equipment and medium 神州医疗科技股份有限公司 2022-09-09 CN disclosed
CN-114996466-A Method and system for establishing medical standard mapping model and using method 神州医疗科技股份有限公司 2022-09-02 CN disclosed
CN-110812442-B Preparation method and application of five-ginseng-astragalus oral solution 湖北威仕生物药业股份有限公司 2022-02-08 CN disclosed