SCHEMBL29372575

SCHEMBL29372575

CCOc1ccn2cc(C3CC3)nc2c1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.45
NPC1 O15118 2/20 0.43
PKM P14618 2/20 0.43
RAB9A P51151 2/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPK1 P28482 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
IRAK4 Q9NWZ3 2/20 0.41
KDM4E B2RXH2 2/20 0.37
POLB P06746 1/20 0.37
HRH3 Q9Y5N1 6/20 0.36
SUV39H2 Q9H5I1 2/20 0.35
MAPT P10636 1/20 0.35
TLR9 Q9NR96 1/20 0.35
TLR7 Q9NYK1 1/20 0.35
ABL1 P00519 1/20 0.34
NOTUM Q6P988 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30259281 0.91 IRAK4 (0.46) PDE10ANPC1PKMRAB9AALDH1A1
SCHEMBL29373194 0.84 NPC1 (0.47) PDE10ANPC1PKMRAB9AKDM4E
SCHEMBL29373916 0.82 PDE10A (0.40) PDE10AIRAK4HRH3SUV39H2
SCHEMBL30259279 0.80 PDE10A (0.42) PDE10ANPC1PKMRAB9AIRAK4
SCHEMBL30427342 0.79 KDM4E (0.43) NPC1PKMRAB9AALDH1A1MAPK1
SCHEMBL25124467 0.74 PDE10A (0.42) PDE10AIRAK4SUV39H2TLR9TLR7
SCHEMBL22234581 0.73 IRAK4 (0.48) PDE10ANPC1PKMRAB9AALDH1A1
SCHEMBL22235013 0.73 IRAK4 (0.48) PDE10ANPC1RAB9AALDH1A1MAPK1
SCHEMBL30259235 0.73 IRAK4 (0.45) NPC1PKMRAB9AALDH1A1MAPK1
Hydrochloric Acid SCHEMBL22235194 0.72 IRAK4 (0.47) PDE10ANPC1RAB9AALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022026935-A1 MULTI-CYCLIC IRAK AND FLT3 INHIBITING COMPOUNDS AND USES THEREOF CHILDREN'S HOSPITAL MEDICAL CENTER (US) 2022-02-03 WO disclosed