SCHEMBL29374201

SCHEMBL29374201

CCOC(=O)c1cc2ccncc2s1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 2/20 0.60
RPS6KA3 P51812 2/20 0.60
CHEK1 O14757 1/20 0.60
AURKA O14965 1/20 0.60
DAPK3 O43293 1/20 0.60
PRKD3 O94806 1/20 0.60
MAP4K4 O95819 1/20 0.60
PAK4 O96013 1/20 0.60
ABL1 P00519 1/20 0.60
RET P07949 1/20 0.60
PIM1 P11309 1/20 0.60
FGFR1 P11362 1/20 0.60
PRKACA P17612 1/20 0.60
FLT1 P17948 1/20 0.60
LTK P29376 1/20 0.60
GRK5 P34947 1/20 0.60
KDR P35968 1/20 0.60
MAPK8 P45983 1/20 0.60
CSNK1A1 P48729 1/20 0.60
CDK8 P49336 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL842776 1.00 GSK3B (0.60) GSK3BRPS6KA3CHEK1AURKADAPK3
SCHEMBL11070341 0.89 CDC7 (0.53) GSK3BRPS6KA3CHEK1AURKADAPK3
SCHEMBL30980399 0.84 CDK8 (0.65) GSK3BRPS6KA3CHEK1AURKADAPK3
SCHEMBL162420 0.84 CDK8 (0.65) GSK3BRPS6KA3CHEK1AURKADAPK3
SCHEMBL4405770 0.79 BCL2L1 (0.57) DYRK1APTPN2MAPTGAAALDH1A1
SCHEMBL29913871 0.79 BCL2L1 (0.57) DYRK1APTPN2MAPTGAAALDH1A1
SCHEMBL13977223 0.79 DYRK1A (0.71) GSK3BRPS6KA3CHEK1AURKADAPK3
SCHEMBL2238245 0.78 PTPN2 (0.60) CDC7DBF4PTPN2MAPTGAA
SCHEMBL8250276 0.78 HDAC1 (0.60) PTPN2MAPTGAAALDH1A1PKM
SCHEMBL26564672 0.78 CHEK1 (0.65) GSK3BRPS6KA3CHEK1AURKADAPK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116730995-B Hydrazide compound, preparation method and application thereof 深圳微芯生物科技股份有限公司 2024-06-25 CN disclosed
CN-109096274-B Biaryl compounds useful in the treatment of human oncological, neurological and immunological diseases 比奥根MA公司 2022-07-01 CN disclosed
CN-108570059-B Compound with PRMT5 inhibitory activity and preparation and application thereof 中国科学院上海药物研究所 2022-02-08 CN disclosed