SCHEMBL29375809

SCHEMBL29375809

COc1cncc(-c2cc3cc(-c4ccc(N5CC6(CCOCC6)C5)nc4)[nH]c3cc2Cl)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 4/20 0.40
KIT P10721 4/20 0.39
ATR Q13535 1/20 0.38
ATRIP Q8WXE1 1/20 0.38
RET P07949 1/20 0.37
KDR P35968 3/20 0.35
CYP17A1 P05093 2/20 0.35
CYP11B1 P15538 2/20 0.35
CYP11B2 P19099 2/20 0.35
ETV6 P41212 1/20 0.35
FYN P06241 2/20 0.35
FGFR1 P11362 2/20 0.34
FGFR2 P21802 2/20 0.34
FGFR3 P22607 2/20 0.34
JAK2 O60674 1/20 0.34
FLT1 P17948 1/20 0.34
FGFR4 P22455 1/20 0.34
LTK P29376 1/20 0.34
FLT4 P35916 1/20 0.34
JAK3 P52333 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21812485 1.00 CNR2 (0.40) CNR2KITATRATRIPRET
SCHEMBL21812349 0.92 CNR2 (0.37) CNR2KITATRATRIPKDR
SCHEMBL29376401 0.92 CNR2 (0.37) CNR2KITATRATRIPKDR
SCHEMBL21812339 0.90 CNR2 (0.49) CNR2KITATRATRIPKDR
SCHEMBL31317860 0.90 CNR2 (0.49) CNR2KITATRATRIPKDR
SCHEMBL21812351 0.88 CYP11B1 (0.37) CNR2KITATRATRIPKDR
SCHEMBL30637807 0.88 CYP11B1 (0.37) CNR2KITATRATRIPKDR
SCHEMBL21812332 0.87 CYP11B1 (0.37) CNR2KITATRATRIPRET
SCHEMBL30637800 0.87 CYP11B1 (0.37) CNR2KITATRATRIPRET
SCHEMBL35210139 0.85 CYP11B1 (0.41) CNR2KITATRATRIPRET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3856736-B1 NOVEL COMPOUNDS AS NADPH OXIDASE INHIBITORS CALLIDITAS THERAPEUTICS SUISSE SA (CH) 2026-05-06 EP claimed
EP-4522162-A1 NOX INHIBITORS FOR USE IN THE TREATMENT OF ALPORT SYNDROME Calliditas Therapeutics Suisse SA (CH) 2025-03-19 EP claimed
US-12202816-B2 Compounds as NADPH oxidase inhibitors CALLIDITAS THERAPEUTICS SUISSE SA (CH) 2025-01-21 US claimed
CN-119212698-A NOX inhibitors for the treatment of Albert syndrome 瑞士商卡利迪塔斯疗法瑞士股份有限公司 2024-12-27 CN claimed
WO-2023217764-A1 NOX INHIBITORS FOR USE IN THE TREATMENT OF ALPORT SYNDROME CALLIDITAS THERAPEUTICS SUISSE SA (CH) 2023-11-16 WO claimed
US-20220033379-A1 NOVEL COMPOUNDS AS NADPH OXIDASE INHIBITORS CALLIDITAS THERAPEUTICS SUISSE SA (CH) 2022-02-03 US claimed
EP-3856736-B1 NOVEL COMPOUNDS AS NADPH OXIDASE INHIBITORS CALLIDITAS THERAPEUTICS SUISSE SA (CH) 2026-05-06 EP disclosed
EP-4522162-A1 NOX INHIBITORS FOR USE IN THE TREATMENT OF ALPORT SYNDROME Calliditas Therapeutics Suisse SA (CH) 2025-03-19 EP disclosed
CN-119212698-A NOX inhibitors for the treatment of Albert syndrome 瑞士商卡利迪塔斯疗法瑞士股份有限公司 2024-12-27 CN disclosed
WO-2023217764-A1 NOX INHIBITORS FOR USE IN THE TREATMENT OF ALPORT SYNDROME CALLIDITAS THERAPEUTICS SUISSE SA (CH) 2023-11-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12202816-B2 Compounds as NADPH oxidase inhibitors CYBB, NOX1, NOX4 CNR2 3184/4885KIT 3394/4885ATR 2916/4885
US-20220033379-A1 NOVEL COMPOUNDS AS NADPH OXIDASE INHIBITORS CYBB, NOX1, NOX4 CNR2 3056/4885KIT 3535/4885ATR 2840/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.