SCHEMBL29376705

SCHEMBL29376705

O=C(O)c1cn2c(cc1=O)-c1ccccc1CC2

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.56
NPC1 O15118 1/20 0.56
MAPT P10636 1/20 0.56
PKM P14618 1/20 0.56
RAB9A P51151 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
SRD5A1 P18405 1/20 0.40
SRD5A2 P31213 1/20 0.40
SERPINE1 P05121 1/20 0.38
ALDH1A1 P00352 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
LMNA P02545 1/20 0.38
HPGD P15428 1/20 0.38
NOTUM Q6P988 1/20 0.38
BCAT2 O15382 1/20 0.36
GAA P10253 1/20 0.36
CTDSP1 Q9GZU7 1/20 0.35
CES1 P23141 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16973636 1.00 KDM4E (0.56) KDM4ENPC1MAPTPKMRAB9A
SCHEMBL21824326 0.92 NPC1 (0.47) KDM4ENPC1MAPTPKMRAB9A
SCHEMBL29521804 0.81 KDM4E (0.46) KDM4ENPC1MAPTPKMRAB9A
SCHEMBL23060734 0.80 KDM4E (0.44) KDM4ENPC1MAPTRAB9ASMN1; SMN2
SCHEMBL29374541 0.80 SMN1; SMN2 (0.40) KDM4ERAB9ASMN1; SMN2ALDH1A1HPGD
SCHEMBL16973490 0.80 SMN1; SMN2 (0.40) KDM4ERAB9ASMN1; SMN2ALDH1A1HPGD
SCHEMBL30137683 0.79 KDM4E (0.42) KDM4EMAPTALDH1A1L3MBTL1
SCHEMBL30607727 0.79 NAPRT (0.37) KDM4ENPC1MAPTPKMRAB9A
SCHEMBL24022985 0.78 ALDH1A1 (0.44) KDM4ENPC1MAPTPKMRAB9A
SCHEMBL21824307 0.77 NOTUM (0.36) KDM4EPKMALDH1A1L3MBTL1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4320117-A2 NOVEL HEPATOSELECTIVE POLYADENYLATING POLYMERASES INHIBITORS AND THEIR METHOD OF USE Baruch S. Blumberg Institute (US) 2024-02-14 EP disclosed
CN-114014854-B Dihydroisoquinoline compound 苏州爱科百发生物医药技术有限公司 2023-04-07 CN disclosed
CN-113999224-B Dihydroisoquinoline compound 苏州爱科百发生物医药技术有限公司 2023-04-07 CN disclosed
WO-2022216552-A2 NOVEL HEPATOSELECTIVE POLYADENYLATING POLYMERASES INHIBITORS AND THEIR METHOD OF USE BARUCH S. BLUMBERG INSTITUTE (US) 2022-10-13 WO disclosed
CN-109715624-B Novel therapeutic agents for the treatment of HBV infection 广州麓鹏制药有限公司 2022-08-16 CN disclosed
CN-114014854-A Dihydroisoquinoline compound 苏州爱科百发生物医药技术有限公司 2022-02-08 CN disclosed
CN-110177785-B Dihydroisoquinoline compound 苏州爱科百发生物医药技术有限公司 2022-02-08 CN disclosed