SCHEMBL29383293

SCHEMBL29383293

CC(C)(C)C#Cc1ccccc1N

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 6/20 0.52
CYP2C9 P11712 4/20 0.52
ALDH1A1 P00352 4/20 0.52
CYP1A2 P05177 3/20 0.52
CYP2C19 P33261 3/20 0.52
KDM4E B2RXH2 2/20 0.52
MAPT P10636 2/20 0.52
SMN1; SMN2 Q16637 2/20 0.52
MEN1 O00255 1/20 0.52
NPC1 O15118 1/20 0.52
HPGD P15428 1/20 0.52
KMT2A Q03164 1/20 0.52
HSD17B10 Q99714 1/20 0.52
PTPN11 Q06124 1/20 0.44
BACE1 P56817 1/20 0.44
CASP3 P42574 1/20 0.43
SENP8 Q96LD8 1/20 0.43
SENP7 Q9BQF6 1/20 0.43
SENP6 Q9GZR1 1/20 0.43
HSP90AA1 P07900 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1258715 1.00 CYP3A4 (0.52) CYP3A4CYP2C9ALDH1A1CYP1A2CYP2C19
SCHEMBL4951135 0.84 BACE1 (0.42) CYP3A4CYP2C9ALDH1A1CYP1A2CYP2C19
SCHEMBL11401297 0.83 CYP3A4 (0.48) CYP3A4CYP2C9ALDH1A1CYP1A2CYP2C19
SCHEMBL29789973 0.83 CYP3A4 (0.48) CYP3A4CYP2C9ALDH1A1CYP1A2CYP2C19
SCHEMBL8536324 0.78 CYP3A4 (0.52) CYP3A4CYP2C9ALDH1A1CYP1A2CYP2C19
SCHEMBL1922269 0.78 CYP3A4 (0.76) CYP3A4CYP2C9ALDH1A1CYP1A2CYP2C19
SCHEMBL618983 0.77 CYP3A4 (0.39) CYP3A4CYP2C9ALDH1A1CYP1A2CYP2C19
SCHEMBL10775408 0.75 ALDH1A1 (0.44) CYP3A4CYP2C9ALDH1A1CYP1A2CYP2C19
SCHEMBL449613 0.75 CYP3A4 (0.58) CYP3A4CYP2C9ALDH1A1CYP1A2CYP2C19
SCHEMBL13597755 0.74 GRM5 (0.42) PTPN11BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110642844-B 3-position indole substituted isobenzofuranone compound and preparation method thereof 郑州大学 2023-03-03 CN disclosed
CN-114031613-A 1- (benzo [ b ] thiophene-7-yl) -indole derivative and synthetic method thereof 湖南第一师范学院 2022-02-11 CN disclosed