SCHEMBL29384604

SCHEMBL29384604

O=C(O)NC1(C(=O)O)CCNCC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.50
KMT2A Q03164 1/20 0.50
CYP1A2 P05177 3/20 0.33
CYP2D6 P10635 1/20 0.33
OPRM1 P35372 1/20 0.31
CYP3A4 P08684 1/20 0.30
GABRP O00591 1/20 0.30
GABRD O14764 1/20 0.30
GABRA1 P14867 1/20 0.30
TSHR P16473 1/20 0.30
GABRB1 P18505 1/20 0.30
GABRG2 P18507 1/20 0.30
GABRB3 P28472 1/20 0.30
GABRA5 P31644 1/20 0.30
GABRA3 P34903 1/20 0.30
GABRA2 P47869 1/20 0.30
GABRB2 P47870 1/20 0.30
GABRA4 P48169 1/20 0.30
GABRE P78334 1/20 0.30
PMP22 Q01453 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18125940 0.83 FFAR3 (0.35)
SCHEMBL21547934 0.83 KDM4E (0.52) KDM4EKMT2ACYP1A2CYP2D6GABRD
SCHEMBL23799317 0.83 KDM4E (0.62) KDM4EKMT2A
SCHEMBL5430016 0.79 KDM4E (0.53) KDM4EKMT2ACYP1A2CYP2D6
SCHEMBL16750982 0.79 KDM4E (0.69) KDM4EKMT2ACYP1A2CYP2D6OPRM1
SCHEMBL18125955 0.78 ALDH1A1 (0.41) CYP1A2
SCHEMBL1957977 0.77 KDM4E (0.55) KDM4EKMT2ACYP1A2CYP2D6CYP3A4
SCHEMBL21082480 0.77 KDM4E (0.42) KDM4EKMT2ATSHR
SCHEMBL10808711 0.76 ALDH1A1 (0.40) CYP1A2
SCHEMBL28045022 0.75 KDM4E (0.53) KDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114940700-A Phenyl propionamide derivative, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2022-08-26 CN disclosed
CN-114349820-A Phenyl propionamide derivative, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2022-04-15 CN disclosed
CN-108290926-B Phenyl propionamide derivative, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2022-02-08 CN disclosed