SCHEMBL29387124

SCHEMBL29387124

CN(C)S(=O)(=O)c1ccc(S(=O)(=O)N2CCC3(CCN(CC(F)(F)F)CC3)c3ccccc32)cc1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 4/20 0.40
NR1I2 O75469 1/20 0.37
RORC P51449 1/20 0.37
NR1H2 P55055 1/20 0.37
NR1H3 Q13133 1/20 0.37
CCR5 P51681 8/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
P2RY1 P47900 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
OPRK1 P41145 1/20 0.34
BRS3 P32247 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25232753 1.00 HTR6 (0.40) HTR6NR1I2RORCNR1H2NR1H3
SCHEMBL26969777 0.93 HTR6 (0.40) HTR6NR1I2RORCNR1H2NR1H3
SCHEMBL26969766 0.90 NPY5R (0.38) HTR6NR1I2RORCNR1H2NR1H3
SCHEMBL25231173 0.86 NPY5R (0.38) NR1I2RORCNR1H2NR1H3P2RY1
SCHEMBL29387287 0.84 CYP3A4 (0.41) CYP3A4CYP2D6CYP2C9CYP2C19MEN1
SCHEMBL25276342 0.84 CYP3A4 (0.41) CYP3A4CYP2D6CYP2C9CYP2C19MEN1
SCHEMBL26969744 0.78 HTR6 (0.40) HTR6P2RY1OPRM1OPRD1OPRK1
SCHEMBL26969727 0.77 NPY5R (0.42) MEN1KMT2A
SCHEMBL26969745 0.76 HDAC1 (0.41) HTR6OPRM1OPRD1
SCHEMBL26969707 0.75 TSHR (0.38) CYP3A4CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4192957-A2 TRPML MODULATORS Casma Therapeutics, Inc. (US) 2023-06-14 EP disclosed
WO-2022032073-A2 TRPML MODULATORS CASMA THERAPEUTICS, INC. (US) 2022-02-10 WO disclosed