Deboxamet

Deboxamet

SCHEMBL29387753

COc1ccc2[nH]c(C)c(CC(=O)NO)c2c1

nearest known ligand 0.74

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C2 P52895 1/20 0.74
MTNR1A P48039 3/20 0.62
MTNR1B P49286 3/20 0.62
HTR1D P28221 2/20 0.58
HTR6 P50406 2/20 0.58
HTR1A P08908 1/20 0.55
SLC6A2 P23975 1/20 0.55
HTR1E P28566 1/20 0.55
HTR7 P34969 1/20 0.55
HTR5A P47898 1/20 0.55
PTPN5 P54829 1/20 0.55
HDAC1 Q13547 7/20 0.54
ALDH1A1 P00352 3/20 0.53
KDM4E B2RXH2 2/20 0.53
MAPT P10636 2/20 0.53
MCL1 Q07820 1/20 0.53
RXFP1 Q9HBX9 1/20 0.53
HDAC3 O15379 1/20 0.53
HDAC4 P56524 1/20 0.53
HDAC7 Q8WUI4 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Deboxamet SCHEMBL186946 1.00 AKR1C2 (0.74) AKR1C2MTNR1AMTNR1BHTR1DHTR6
SCHEMBL8270880 0.90 AKR1C2 (0.74) AKR1C2MTNR1AMTNR1BHTR1DHTR6
SCHEMBL8110763 0.87 AKR1C2 (0.70) AKR1C2MTNR1AMTNR1BHTR1DHTR6
SCHEMBL8401335 0.87 AKR1C2 (0.70) AKR1C2MTNR1AMTNR1BHTR1DHTR6
SCHEMBL30604527 0.86 AKR1C2 (0.78) AKR1C2MTNR1AMTNR1BHTR1DHTR6
SCHEMBL6825151 0.86 AKR1C2 (0.78) AKR1C2MTNR1AMTNR1BHTR1DHTR6
SCHEMBL7960856 0.85 AKR1C2 (0.67) AKR1C2MTNR1AMTNR1BHTR1DHTR6
Deschlorobenzoyl Indomethacin SCHEMBL454792 0.85 AKR1C2 (1.00) AKR1C2MTNR1AMTNR1BHTR1DHTR6
SCHEMBL10205891 0.85 AKR1C2 (0.80) AKR1C2MTNR1AMTNR1BHTR1DHTR6
SCHEMBL4825986 0.85 AKR1C2 (0.57) AKR1C2MTNR1AMTNR1BHDAC1HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116157404-A Heteroaryl substituted spiropiperidinyl derivatives and pharmaceutical uses thereof 诺华股份有限公司 2023-05-23 CN disclosed
CN-114884565-B Large-scale low-orbit satellite network topology optimization method based on communication performance constraint 南京大学 2023-05-09 CN disclosed
CN-114884565-A Communication performance constraint-based large-scale low-orbit satellite network topology optimization method 南京大学 2022-08-09 CN disclosed
CN-114716544-A Complement component C5 antibody 阿勒根公司 2022-07-08 CN disclosed
US-20220047505-A1 Controlled Absorption Water-Soluble Pharmaceutically Active Organic Compound Formulation for Once-Daily Administration STI PHARMA, LLC (US) 2022-02-17 US disclosed