SCHEMBL29388181

SCHEMBL29388181

CC(=O)c1ccc(N)c(F)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.61
HDAC6 Q9UBN7 1/20 0.61
PRKCI P41743 1/20 0.52
CREBBP Q92793 1/20 0.47
ALDH1A1 P00352 1/20 0.46
CES2 O00748 1/20 0.43
CES1 P23141 1/20 0.43
SLC6A5 Q9Y345 1/20 0.43
NPC1 O15118 2/20 0.42
MAPT P10636 2/20 0.42
RAB9A P51151 2/20 0.42
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA4 P22748 1/20 0.42
CA6 P23280 1/20 0.42
CA5A P35218 1/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42
CA14 Q9ULX7 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL478933 1.00 HDAC1 (0.61) HDAC1HDAC6PRKCICREBBPALDH1A1
SCHEMBL5332682 0.85 HDAC1 (0.47) HDAC1HDAC6PRKCICREBBPALDH1A1
SCHEMBL935912 0.83 PRKCI (0.56) HDAC1HDAC6PRKCICREBBPALDH1A1
SCHEMBL863794 0.83 HDAC1 (0.66) HDAC1HDAC6ALDH1A1CES2CES1
SCHEMBL29367661 0.81 HDAC1 (0.63) HDAC1HDAC6ALDH1A1CES2CES1
SCHEMBL1627106 0.81 HDAC1 (0.63) HDAC1HDAC6ALDH1A1CES2CES1
SCHEMBL97816 0.81 HDAC1 (0.63) HDAC1HDAC6ALDH1A1CES2CES1
SCHEMBL4453036 0.81 MAPT (0.61) HDAC1HDAC6ALDH1A1MAPTRAB9A
SCHEMBL29669896 0.80 CES2 (0.67) CES2CES1NPC1MAPTRAB9A
SCHEMBL75801 0.80 CES2 (0.67) CES2CES1NPC1MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3560926-B1 6-AMINO-7,9-DIHYDRO-8H-PURIN-8-ONE COMPOUNDS AS BRK INHIBITORS ONO PHARMACEUTICAL CO (JP) 2022-02-23 EP disclosed