SCHEMBL29403449

SCHEMBL29403449

FC(F)c1ccc2cccnc2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.53
HTT P42858 3/20 0.53
CASP1 P29466 2/20 0.53
MEN1 O00255 1/20 0.53
CASP7 P55210 1/20 0.53
KMT2A Q03164 1/20 0.53
CYP1A2 P05177 1/20 0.53
CYP2C19 P33261 1/20 0.53
NR4A2 P43354 1/20 0.53
OGA O60502 3/20 0.52
CYP3A4 P08684 4/20 0.48
CYP2D6 P10635 2/20 0.48
SLC6A2 P23975 1/20 0.48
SLC6A4 P31645 1/20 0.48
SLC6A3 Q01959 1/20 0.48
NPC1 O15118 2/20 0.42
POLB P06746 1/20 0.42
RAB9A P51151 1/20 0.42
PDGFRB P09619 1/20 0.42
PDGFRA P16234 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17785872 1.00 ALDH1A1 (0.53) ALDH1A1HTTCASP1MEN1CASP7
SCHEMBL14322835 0.85 NPC1 (0.57) ALDH1A1HTTCASP1MEN1KMT2A
SCHEMBL903412 0.85 ALDH1A1 (0.58) ALDH1A1HTTCASP1MEN1CASP7
SCHEMBL30644683 0.81 UGT2B7 (0.56) ALDH1A1HTTCASP1MEN1CASP7
SCHEMBL17541507 0.81 UGT2B7 (0.56) ALDH1A1HTTCASP1MEN1CASP7
SCHEMBL30644592 0.81 ALDH1A1 (0.55) ALDH1A1HTTCASP1MEN1CASP7
SCHEMBL17541523 0.81 ALDH1A1 (0.55) ALDH1A1HTTCASP1MEN1CASP7
SCHEMBL11873906 0.81 HTT (0.58) ALDH1A1HTTCASP1MEN1CASP7
Hydrochloric Acid SCHEMBL27757951 0.80 ALDH1A1 (0.53) ALDH1A1HTTCASP1MEN1CASP7
SCHEMBL12386875 0.79 ALDH1A1 (0.51) ALDH1A1HTTCASP1MEN1CASP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116507333-B Cyclic AMP response element binding protein (CBP) and/or 300KDA adenovirus E1A binding protein (P300) degrading compounds and methods of use 上海睿跃生物科技有限公司 2025-05-09 CN disclosed
CN-119330963-A Cyclic AMP response element binding protein (CBP) and/or 300KDA adenovirus E1A binding protein (P300) degrading compounds and methods of use 上海睿跃生物科技有限公司 2025-01-21 CN disclosed
CN-112165944-B Imidazopiperazine inhibitors of transcriptional activator proteins 德州大学系统董事会 2024-04-09 CN disclosed
CN-116507333-A Cyclic AMP response element binding protein (CBP) and/or 300KDA adenovirus E1A binding protein (P300) degrading compounds and methods of use 上海睿跃生物科技有限公司 2023-07-28 CN disclosed
EP-4157888-A1 MODIFIED PROTEINS AND PROTEIN DEGRADERS Cullgen (Shanghai), Inc. (CN) 2023-04-05 EP disclosed
CN-115028617-A Heterocyclic inhibitors of CBP/EP300 and their use in the treatment of cancer 基因泰克公司 2022-09-09 CN disclosed
CN-109476641-B Heterocyclic inhibitors of CBP/EP300 and their use in the treatment of cancer 基因泰克公司 2022-07-05 CN disclosed
WO-2022042707-A1 CYCLIC-AMP RESPONSE ELEMENT BINDING PROTEIN (CBP) AND/OR ADENOVIRAL E1A BINDING PROTEIN OF 300 KDA (P300) DEGRADATION COMPOUNDS AND METHODS OF USE CULLGEN (SHANGHAI) , INC. (CN) 2022-03-03 WO disclosed