SCHEMBL2941010

SCHEMBL2941010

CCOc1cnccc1C(C)C1(C(C)c2ccncc2OCC)NC(=O)N(c2ccc(OC(F)(F)F)cc2)C1=O

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.36
POLB P06746 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
GAA P10253 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CXCR3 P49682 8/20 0.36
AR P10275 1/20 0.33
ABL1 P00519 1/20 0.33
LIPE Q05469 1/20 0.33
CACNA2D1 P54289 1/20 0.33
LMNA P02545 1/20 0.33
CCR6 P51684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6173690 0.90 CYP3A4 (0.41) CYP3A4POLBL3MBTL1GAACYP2C9
SCHEMBL6172003 0.87 ALDH1A1 (0.37) CYP3A4POLBL3MBTL1GAACYP2C9
SCHEMBL6173429 0.86 POLB (0.41) CYP3A4POLBL3MBTL1GAACYP2C9
SCHEMBL6177840 0.86 IGF1R (0.43) AR
SCHEMBL6174774 0.85 SLC5A1 (0.40) CYP3A4POLBL3MBTL1GAACYP2C9
SCHEMBL6170701 0.85 IGF1R (0.37) CYP3A4GAACYP2C9CYP2C19ALDH1A1
SCHEMBL6170901 0.85 CYP3A4 (0.35) CYP3A4POLBL3MBTL1GAACYP2C9
SCHEMBL6173440 0.85 CYP3A4 (0.38) CYP3A4POLBL3MBTL1GAACYP2C9
SCHEMBL6175704 0.85 POLB (0.36) CYP3A4POLBL3MBTL1GAACYP2C9
SCHEMBL6173276 0.83 CYP3A4 (0.35) CYP3A4POLBL3MBTL1GAACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1599464-B1 NOVEL CYCLIC UREA DERIVATIVES, PREPARATION METHOD THEREOF AND PHARMACEUTICAL USE OF SAME AS KINASE INHIBITORS AVENTIS PHARMA SA (FR) 2010-09-22 EP disclosed