SCHEMBL29414458

SCHEMBL29414458

CCN1CCN(Cc2ccc(Nc3ncc(F)c(-c4ccc5nc(C)c(C)nc5c4)n3)nc2)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CDK6 Q00534 15/20 1.00
DYRK2 Q92630 5/20 0.77
CCND3 P30281 8/20 0.71
CCND1 P24385 6/20 0.71
CDK4 P11802 6/20 0.71
CDK1 P06493 5/20 0.68
CCNA2 P20248 5/20 0.68
CCNE2 O96020 4/20 0.68
CDK2 P24941 4/20 0.68
PIM1 P11309 2/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28591508 1.00 CDK6 (1.00) CDK6DYRK2CCND3CCND1CDK4
SCHEMBL28595397 0.91 CDK6 (1.00) CDK6DYRK2CCND3CCND1CDK4
SCHEMBL29414464 0.91 CDK6 (1.00) CDK6DYRK2CCND3CCND1CDK4
SCHEMBL29379886 0.90 CDK6 (0.82) CDK6DYRK2CCND3CCND1CDK4
SCHEMBL28595830 0.90 CDK6 (0.82) CDK6DYRK2CCND3CCND1CDK4
Hydrochloric Acid SCHEMBL28592444 0.90 CDK6 (0.81) CDK6DYRK2CCND3CCND1CDK4
Hydrochloric Acid SCHEMBL29414470 0.90 CDK6 (0.81) CDK6DYRK2CCND3CCND1CDK4
SCHEMBL26447899 0.87 DYRK2 (1.00) CDK6DYRK2CCND3CCND1CDK4
SCHEMBL32677350 0.87 DYRK2 (1.00) CDK6DYRK2CCND3CCND1CDK4
SCHEMBL29754375 0.87 DYRK2 (0.87) CDK6DYRK2CCND3CCND1CDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113135898-B Anticancer quinoxaline pyrimidine amine heterocyclic compound and preparation method and application thereof 中国药科大学 2022-02-11 CN disclosed