SCHEMBL28595397

SCHEMBL28595397

Cc1nc2ccc(-c3nc(Nc4ccc(CN5CCN(C(C)C)CC5)cn4)ncc3F)cc2nc1C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CDK6 Q00534 13/20 1.00
DYRK2 Q92630 7/20 0.78
CCND1 P24385 4/20 0.72
CDK4 P11802 4/20 0.63
CDK1 P06493 2/20 0.60
CCNA2 P20248 2/20 0.60
CCND3 P30281 2/20 0.60
PIM1 P11309 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29414464 1.00 CDK6 (1.00) CDK6DYRK2CCND1CDK4CDK1
SCHEMBL28592563 0.91 CDK6 (1.00) CDK6DYRK2CCND1CDK4CDK1
SCHEMBL29414498 0.91 CDK6 (1.00) CDK6DYRK2CCND1CDK4CDK1
SCHEMBL29414458 0.91 CDK6 (1.00) CDK6DYRK2CCND1CDK4CDK1
SCHEMBL28591508 0.91 CDK6 (1.00) CDK6DYRK2CCND1CDK4CDK1
SCHEMBL29230288 0.88 DYRK2 (1.00) CDK6DYRK2CCND1CDK4
SCHEMBL30917869 0.88 DYRK2 (1.00) CDK6DYRK2CCND1CDK4
Hydrochloric Acid SCHEMBL28592444 0.87 CDK6 (0.81) CDK6DYRK2CCND1CDK4CDK1
Hydrochloric Acid SCHEMBL29414470 0.87 CDK6 (0.81) CDK6DYRK2CCND1CDK4CDK1
SCHEMBL29754496 0.87 DYRK2 (0.83) CDK6DYRK2CCND1CDK4CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113135898-B Anticancer quinoxaline pyrimidine amine heterocyclic compound and preparation method and application thereof 中国药科大学 2022-02-11 CN disclosed
CN-113135898-A Anticancer quinoxaline pyrimidine amine heterocyclic compound and preparation method and application thereof 中国药科大学 2021-07-20 CN disclosed