SCHEMBL29416645

SCHEMBL29416645

COc1cc(O)c(C(=O)/C=C/c2ccc(O)c(O)c2)cc1OC

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.71
CYP3A4 P08684 3/20 0.70
CYP1A2 P05177 1/20 0.70
CYP2D6 P10635 1/20 0.70
CYP2C9 P11712 1/20 0.70
CYP2C19 P33261 1/20 0.70
CHRNA7 P36544 1/20 0.65
PDE4A P27815 1/20 0.65
PDE4B Q07343 1/20 0.65
PDE4C Q08493 1/20 0.65
PDE4D Q08499 1/20 0.65
MAPT P10636 2/20 0.64
SMN1; SMN2 Q16637 2/20 0.64
AR P10275 1/20 0.64
MEN1 O00255 1/20 0.64
ALDH1A1 P00352 1/20 0.64
TP53 P04637 1/20 0.64
HPGD P15428 1/20 0.64
ALOX15 P16050 1/20 0.64
ALOX12 P18054 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28678909 1.00 MAOB (0.71) MAOBCYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL19086304 0.90 ABCG2 (0.78) MAOBCYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL19086305 0.90 ABCG2 (0.78) MAOBCYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL25223496 0.86 CYP3A4 (0.67) MAOBCYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL25223485 0.86 CYP3A4 (0.66) MAOBCYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL25238512 0.86 ACHE (0.81) MAOBCYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL25204409 0.85 CYP3A4 (0.65) MAOBCYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL25266095 0.84 ABCG2 (0.76) MAOBMAPTMAPK1KMT2AABCG2
SCHEMBL25239854 0.84 ACHE (0.81) CYP3A4CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL31233136 0.84 ABCG2 (0.76) MAOBMAPTMAPK1KMT2AABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114105753-A Fisetin derivative and application thereof in preparation of anti-inflammatory drugs 温州医科大学 2022-03-01 CN claimed
CN-114105753-B Fisetin derivative and application thereof in preparation of anti-inflammatory drugs 温州医科大学 2024-02-20 CN disclosed
CN-114105753-A Fisetin derivative and application thereof in preparation of anti-inflammatory drugs 温州医科大学 2022-03-01 CN disclosed