SCHEMBL29426430

SCHEMBL29426430

O=C(O)/C(=C/c1ccccc1)c1cccc2ccccc12

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.80
CYP3A4 P08684 3/20 0.80
CYP2D6 P10635 3/20 0.80
CYP2C9 P11712 2/20 0.80
CYP2C19 P33261 2/20 0.80
AKR1C2 P52895 1/20 0.64
KMT2A Q03164 2/20 0.60
NR4A1 P22736 1/20 0.56
NR4A2 P43354 1/20 0.56
NR4A3 Q92570 1/20 0.56
AKR1C1 Q04828 1/20 0.55
CDC25B P30305 1/20 0.50
MMP3 P08254 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
MAPT P10636 2/20 0.47
NPSR1 Q6W5P4 1/20 0.47
PTPN1 P18031 1/20 0.46
PLK1 P53350 1/20 0.46
CYP1A1 P04798 1/20 0.44
CYP1B1 Q16678 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11435631 1.00 CYP1A2 (0.80) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL6563634 0.87 CYP1A2 (0.78) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL6563624 0.87 CYP1A2 (0.78) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
Naphthoic Acid SCHEMBL27147498 0.86 AKR1C1 (0.65) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL17541843 0.85 CYP1A2 (0.61) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL27972507 0.85 CYP1A2 (0.61) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL11670349 0.85 CYP1A2 (0.64) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL28216150 0.85 CYP1A2 (0.64) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL11670351 0.85 CYP1A2 (0.64) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL1646802 0.83 AKR1C1 (0.69) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022048922-A1 SUBSTITUTED VICINAL DIAMINE COMPOUNDS AND THEIR USE IN THE TREATMENT, AMELIORATION OR PREVENTION OF PAIN Friedrich-Alexander-Universität Erlangen-Nürnberg (DE) 2022-03-10 WO disclosed