SCHEMBL29426488

SCHEMBL29426488

COC(=O)Cn1nc(I)c2ccc(Br)cc2c1=O

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.49
CASP3 P42574 2/20 0.46
NLRP3 Q96P20 1/20 0.43
CDK1 P06493 2/20 0.40
MCL1 Q07820 1/20 0.40
KDM4E B2RXH2 3/20 0.39
LMNA P02545 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
HTT P42858 1/20 0.39
KMT2A Q03164 1/20 0.39
FPR1 P21462 2/20 0.39
FPR2 P25090 2/20 0.39
EGFR P00533 1/20 0.38
HSD17B10 Q99714 1/20 0.38
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26732573 1.00 TSHR (0.49) TSHRCASP3NLRP3CDK1MCL1
SCHEMBL26732572 0.95 TSHR (0.52) TSHRCASP3NLRP3CDK1MCL1
SCHEMBL29426511 0.86 TSHR (0.48) TSHRCASP3NLRP3MCL1KDM4E
SCHEMBL26733144 0.86 TSHR (0.48) TSHRCASP3NLRP3MCL1KDM4E
SCHEMBL24257391 0.86 TSHR (0.53) TSHRCASP3NLRP3MCL1KDM4E
SCHEMBL29426475 0.86 TSHR (0.53) TSHRCASP3NLRP3MCL1KDM4E
SCHEMBL29426501 0.85 TSHR (0.47) TSHRCASP3NLRP3CDK1MCL1
SCHEMBL29426497 0.85 TSHR (0.47) TSHRCASP3NLRP3CDK1MCL1
SCHEMBL29426519 0.85 TSHR (0.47) TSHRCASP3NLRP3CDK1MCL1
SCHEMBL26732856 0.85 TSHR (0.47) TSHRCASP3NLRP3CDK1MCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4196125-A1 COMPOUNDS, COMPOSITIONS AND METHODS Denali Therapeutics Inc. (US) 2023-06-21 EP disclosed
WO-2022036204-A1 COMPOUNDS, COMPOSITIONS AND METHODS DENALI THERAPEUTICS INC. (US) 2022-02-17 WO disclosed