SCHEMBL2942862

SCHEMBL2942862

CCCCCc1cccc(NC(N)=S)c1C(=O)c1cc2cccnc2o1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.40
CYP3A4 P08684 2/20 0.40
TRPV1 Q8NER1 3/20 0.37
MAPK1 P28482 2/20 0.36
MAPT P10636 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
TLR8 Q9NR97 1/20 0.35
BID P55957 3/20 0.34
MCL1 Q07820 3/20 0.34
BCL2L1 Q07817 2/20 0.34
BAK1 Q16611 2/20 0.34
KAT8 Q9H7Z6 2/20 0.34
PPARA Q07869 2/20 0.34
PPARG P37231 1/20 0.34
EP300 Q09472 1/20 0.34
KAT2A Q92830 1/20 0.34
KAT2B Q92831 1/20 0.34
KAT5 Q92993 1/20 0.34
SAE1 Q9UBE0 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2945223 0.86 PTPN1 (0.40) CYP1A2CYP3A4MAPK1MAPTNPSR1
SCHEMBL4361608 0.86 HDAC3 (0.45) MAPK1MAPTNPC1RAB9AKDM4E
SCHEMBL2942857 0.81 CYP1A2 (0.39) CYP1A2CYP3A4MAPK1MAPTNPSR1
SCHEMBL2942290 0.80 NPC1 (0.43) MAPTNPSR1NPC1RAB9AALDH1A1
SCHEMBL2945216 0.79 CYP1A2 (0.38) CYP1A2CYP3A4MAPTNPC1RAB9A
SCHEMBL2918621 0.76 CYP1A2 (0.38) CYP1A2CYP3A4TRPV1MAPK1MAPT
SCHEMBL2915541 0.76 CYP1A2 (0.41) CYP1A2CYP3A4MAPK1MAPTNPSR1
SCHEMBL13175642 0.72 MAPT (0.52) TRPV1MAPK1MAPTNPSR1RXFP1
SCHEMBL4357780 0.70 MAOB (0.52) MAPK1MAPTNPSR1NPC1RAB9A
SCHEMBL11405552 0.69 L3MBTL1 (0.56) CYP1A2CYP3A4TRPV1MAPK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1709047-B1 AZABENZOFURAN SUBSTITUTED THIOUREAS AS INHIBITORS OF VIRAL REPLICATION ACHILLION PHARMACEUTICALS INC (US) 2010-09-01 EP claimed